BTRX 335140 CAS 2244614-14-8

BTRX 335140 CAS 2244614-14-8

Khoom npe: BTRX-335140
Synonym: CYM-53093; Navacaprant
CAS Nr .: 2244614-14-8
EINECS NO.:/
Cov mis mos molecular: C25H32FN5O2
Purity & Qib: 99%; Qib tshuaj
Cim: Dawb hmoov
Cov qauv dawb: Muaj
Tshuag: Hauv Tshuag
Warehouse: USA/EU/AU Warehouse
MOQ & Pob: 1g; Pob raws li xav tau
Shipping: Kev nyab xeeb thiab xa khoom sai
Lub Sijhawm Lead: 5-10 hnub
Khw & Txee lub neej: Txias & qhuav qhov chaw; 24 hli
Xa kev nug
Hauj lwm lawm
 
 

Khoom piav qhia

BTRX 335140 CAS 2244614-14-8

BTRX 335140 CAS 2244614-14-8, tseem hu ua Navacaprant, feem ntau yog tsom rau lub hauv paus paj hlwb lub luag haujlwm hauv kev xav thiab kev paub txog kev tswj hwm. Cov tshuaj no ua haujlwm nrog kev xaiv siab ntawm κ-opioid receptors, nthuav tawm muaj zog affinity rau nws lub hom phiaj qhov chaw, thaum tso tawm tsis tshua muaj ntoo khaub lig- ua haujlwm nrog μ thiab δ-opioid receptors. Yog li ntawd, nws muaj qhov txiaj ntsig tseem ceeb hauv nws cov txheej txheem ntawm kev ua haujlwm, zam qhov kev pheej hmoo tsis zoo uas feem ntau cuam tshuam nrog cov tshuaj muaj feem cuam tshuam. Nws cov txheej txheem ntawm kev ua haujlwm feem ntau suav nrog kev tswj cov dynorphin-KOR teeb liab qhov system, txhim kho kev ua haujlwm ntawm cov nqi zog, kev txhawb siab, thiab kev tswj hwm kev xav hauv lub hlwb, tshwj xeeb tshaj yog tsom rau qhov tshwm sim tseem ceeb xws li kev nyuaj siab thiab tsis txaus siab. Nws muaj cov ntshav zoo- lub hlwb thaiv kev nkag mus thiab cov yam ntxwv ntawm kev nqus tau ruaj khov, tswj cov nyhuv ruaj khov nrog ib zaug - kev tswj hwm txhua hnub.

Nyob rau hauv kev tshawb fawb soj ntsuam thaum ntxov, BTRX-335140 tau pom cov txiaj ntsig zoo thiab kev ua siab ntev, dhau los ua qhov kev xav tau zoo tshaj plaws hauv kev tshawb fawb hauv cheeb tsam ntawm kev ua haujlwm. Txawm hais tias cov kev tshawb fawb tseem ceeb tom qab tsis tau ua tiav cov hom phiaj xav tau, cuam tshuam nws txoj kev nce qib hauv cov kev taw qhia tseem ceeb, cov khoom tseem tab tom tshawb nrhiav hauv thaj chaw ntawm kev puas siab puas ntsws bipolar thiab muab cov ntaub ntawv tseem ceeb thiab kev paub txog kev tshawb fawb thiab kev loj hlob ntawm cov txheej txheem zoo sib xws, uas yog qhov tseem ceeb hauv kev tshawb fawb thiab kev loj hlob ntawm cov molecules me me nrog lub hauv paus paj hlwb kev ua ub no.

BTRX 335140 CAS 2244614-14-8

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

COA

 

Kev sim Specifications Cov txiaj ntsig
Qhov tshwm sim Dawb hmoov Ua raws
Specification 98% Ua raws
tsw Yam ntxwv Ua raws
Particle loj 100% dhau 80 mesh Ua raws
Cov hlau hnyav
Total Heavy metals Tsawg dua lossis sib npaug li 10ppm Ua raws
Microbial
Tag nrho microbacterial suav Tsawg dua lossis sib npaug li 1000cfu / g Ua raws
Poov & Mould Tsawg dua lossis sib npaug li 100cfu / g Ua raws
Escherichia Coli muaj nyob Tsis zoo Ua raws
Salmonella Tsis zoo Ua raws
Staphylococcus Tsis zoo Ua raws
Xaus Ua raws li kev lag luam specification

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

MF of BTRX-335140

Cov roj formula: C25H32FN5O2
Molecular Luj: 453.55
InChIKey CQOJHAJWCDJEAT-UHFFFAOYSA-N
SMILES Ccc1cc(F)c2nc(N3CCC(NC4CCOCC4)CC3)c(-c3nc(C)no3)c(C)c2c1
Qhov tsos: Khoom
Cia txias: 2-8 degree

Cov ntsiab lus tseem ceeb ntawm BTRX 335140 CAS 2244614-14-8

 

Lub luag haujlwm tseem ceeb ntawm kev ua ntawm BTRX-335140 (Navacaprant) yog xaiv los khi rau thiab thaiv kev ua haujlwm ntawm κ-opioid receptors (KOR) hauv nruab nrab paj hlwb, inhibiting kev sib kis ntawm dynorphin-txog txoj hauv kev. Qhov no txo ​​qis cov nyhuv inhibitory ntawm cov neurotransmitter systems xws li dopamine, tswj cov neural circuits hauv lub hlwb ntsig txog kev xav, nqi zog kev xav, kev txhawb siab, thiab kev ntxhov siab. Cov molecule no muaj kev sib raug zoo thiab kev xaiv rau κ-opioid receptors, thaum pom tias muaj kev sib raug zoo tsis muaj zog rau lwm hom opioid receptors, yog li nws qhov kev txiav txim siab ntau dua thiab tsis tshua muaj kev cuam tshuam los yog ua siab ntev. Vim nws cov ntshav-hlwb thaiv kev nkag mus thiab nqus tau zoo, nws feem ntau yog siv hauv kev tshawb fawb ntsig txog kev tswj hwm lub siab, tsom mus rau cov kev tshwm sim xws li kev nyuaj siab, tsis txaus siab, thiab anhedonia, thiab tau tshawb nrhiav hauv chaw kho mob xws li mob hnyav thiab kev puas siab puas ntsws bipolar.

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

BTRX 335140 CAS 2244614-14-8

vim li cas xaiv peb

 
Peb ua raws li lub hauv paus ntsiab lus ntawm "tus neeg siv khoom ua ntej, kev ua siab ncaj ua ntej", thiab ib txwm muab cov neeg siv khoom nrog cov khoom zoo thiab muaj txiaj ntsig zoo thiab - cov kev pabcuam zoo. Xaiv kev ncaj ncees. Xaiv lub neej noj qab nyob zoo!
 
Nrog rau peb cov kev siv zog tas mus li thiab kev pabcuam zoo, peb cia siab tias yuav tsim kom muaj kev koom tes ntev - thiab kev loj hlob zoo nrog cov neeg siv khoom thiab muab sijhawm rau peb. Peb ntseeg tias peb yuav txaus siab rau koj nrog thawj -chav kawm zoo, nyab xeeb thiab xa khoom sai thiab txaus siab tom qab- kev muag khoom.

 

Peb lub Hoobkas

 

BTRX 335140 CAS 2244614-14-8

BTRX 335140 CAS 2244614-14-8

 

Pob

 

BTRX 335140 CAS 2244614-14-8

 

Shipping Txoj Kev

 

Tsheb thauj mus los

Shipping txoj kev

Cargo hnyav xav tau

Qhov zoo

3-7 hnub

DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD,
UPS, USPS, FedEx, TNT, EMS

Haum rau qis dua 50kg.
International qhov rooj rau qhov rooj nthuav qhia

Peb muaj warehouses nyob rau hauv lub teb chaws Yelemees thiab California, teb chaws USA, thiab cov neeg muas zaub nyob rau hauv cov teb chaws Europe thiab America yuav txaus siab rau xa cov khoom ncaj qha los ntawm ob qhov chaw.

7-15 hnub

Los ntawm Cua

Haum rau ntau tshaj 50kg.
ceev thiab pheej yig dua rau kev txiav txim loj

15-60 hnub

Los ntawm Hiav Txwv

Haum rau ntau tshaj 500kg.
Kev xa khoom pheej yig tshaj plaws

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

FAQ

 

 

01. Dab tsi yog qhov tseem ceeb ntawm BTRX 335140 CAS 2244614-14-8 rau kev tshawb fawb kev lag luam?

Raws li tus neeg sawv cev molecule tsom rau κ-opioid receptor, nws muab cov ntaub ntawv kho mob tseem ceeb rau kev tswj hwm lub paj hlwb hauv nruab nrab thiab muab cov ntaub ntawv tseem ceeb rau kev txhim kho kev taw qhia thiab kev tshuaj ntsuam xyuas ntawm cov molecules tom ntej nrog cov txheej txheem zoo sib xws.

02. Qhov kev tshawb fawb tsom mus rau qhov twg BTRX 335140 CAS 2244614-14-8 txog tam sim no?

Tom qab kev tshawb fawb thawj zaug hauv nws qhov kev taw qhia thawj zaug ua tsis tau raws li qhov kev cia siab, qhov kev tshawb fawb tsom tau maj mam hloov mus rau thaj tsam ntawm kev puas siab puas ntsws bipolar -txog kev puas siab puas ntsws, thiab txuas ntxiv tshawb xyuas cov pej xeem meej dua thiab cov tswv yim tswj hwm kev sib koom ua ke.

03. Kuv tuaj yeem yuav BTRX 335140 CAS 2244614-14-8 qhov twg?

Koj tuaj yeem tiv tauj tus email chaw nyob hauv qab no:sales4@faithfulbio.com
 
Tsis lees paub: Tag nrho cov khoom lag luam (tsis yog- cov khoom siv kho mob) cov duab raug coj los ua zoo, tab sis vim yog lub zog ntawm lub teeb (lub sijhawm sib txawv, lub teeb tom qab sib txawv), txoj kev tua, cov khoom siv sib txawv thiab lwm yam, tej zaum yuav muaj qee qhov sib txawv ntawm daim duab thiab cov xim tiag tiag, cov xim ntawm cov khoom, thov coj cov nyhuv tiag tiag, xim txawv ntawm cov khoom tsis yog qhov teeb meem zoo.
 
Nco tseg: Nco ntsoov sab laj nrog tus kws kho mob uas tsim nyog ua ntej noj cov tshuaj tshiab. Cov khoom no tsis yog tsim los kuaj xyuas, kho, kho lossis tiv thaiv txhua yam kab mob.Thaum lub sijhawm yuav khoom, tus neeg yuav khoom thoob ntiaj teb pom zoo xav tias muaj kev pheej hmoo ntawm txhua yam khoom tuaj txog. Peb tsis tuaj yeem hloov cov khoom ploj lossis raug kaw. Ua ntej xa cov khoom, koj yuav tsum paub meej tias koj pom zoo rau cov nqe lus no.Qhov no tsuas yog kev pom zoo koob tshuaj raws li peb tus kheej kev paub thiab cov ntaub ntawv pov thawj. Peb pom zoo kom koj ua koj tus kheej kev tshawb fawb ua ntej siv cov khoom no.
 
Nqe lus:Cov khoom no tsuas yog siv rau kev tshawb fawb tshawb fawb, thiab qhov tshwm sim ntawm lwm yam kev siv tsis muaj lub luag haujlwm.

 

Cim npe nrov: btrx 335140 cas 2244614-14-8, Tuam Tshoj, lwm tus neeg, manufacturers, hoobkas, customized, lag luam wholesale, yuav, nqe, tej, ntshiab, tsim, luv nqi, kev muag, Tshuag, dawb qauv, raw hmoov, raw khoom, ua nyob rau hauv Suav teb