99% CB-03-01 hmoovyog hu ua CB rau luv thiab tom qab lub npeBreezula, tab sis nws lub npe tshuaj kuj hu uaClascoterone. Nws yog ib qho tshuaj tiv thaiv androgen sab nraud nrog ob peb cov kev mob tshwm sim thiab tam sim no nyob rau theem kho mob.
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| CB-03-01 hmoov | Clascoterone Cov Qauv Qauv |
Khoom siv
Cosmo Pharmaceuticals, lub tuam txhab tshuaj Italian, ua kev tshawb fawb soj ntsuam ntawm nws, uas yog siv rau sab nraud siv los kho pob txuv, hirsutism, thiab plaub hau poob. Nws yog ib qho tshuaj rau kev kho mob ntawm cov txiv neej cov plaub hau poob nyob rau hauv lub sij hawm luv luv nyob rau hauv lub neej yav tom ntej, thiab feem ntau yuav lwm txoj rau finasteride,
Cosmo pharmaceuticals tso tawm cov ntaub ntawv tshawb xyuas ib ntus ntawm theem II kev soj ntsuam kev sim ntawmBreezula, uas yog lub hom phiaj tseem ceeb ntawm kev txiav txim siab ntau npaum li cas thiab kev sim ntxiv rau kev ua tau zoo thiab kev nyab xeeb ntawm cov tshuaj.
Cov koob tshuaj ntawm qhov kev sim no feem ntau suav nrog 2.5% ob zaug hauv ib hnub, 5% ob zaug hauv ib hnub, 7.5% ob zaug hauv ib hnub, 7.5% ib hnub ib zaug, thiab pawg tswj kev sim.
Raws li cov ntaub ntawv ntsuam xyuas, peb tuaj yeem paub tias thaj chaw coated nrog CB tau ua kom zoo dua ntawm cov plaub hau thiab qhov kev ntsuam xyuas ntawm cov plaub hau. Nyob rau tib lub sijhawm, hauv kev sim, peb tuaj yeem pom tias qhov koob tshuaj zoo tshaj plaws yog 7.5% CB, uas yog siv ob zaug ib hnub.
Nyob rau tib lub sijhawm, raws li kev tshawb fawb xaus,99% ntawm CB-03-01 hmoovrau kev siv sab nraud yeej tsis nkag mus rau tib neeg cov ntshav rau cov metabolism, yog li nws yuav tsis cuam tshuam nrog cov qib ntawm cov tshuaj hormones hauv tib neeg lub cev, tshwj xeeb tshaj yog testosterone. Tsis muaj kev phiv ntawm qhov nam no tau pom nyob rau hauv cov txheej txheem ntawm kev sim tshuaj.
Hauv qhov kev sim, cov tshuaj tiv thaiv ntawm daim tawv nqaij hauv zos tau muab faib ua me me, thiab tsis pom muaj qhov tshwm sim ntawm daim tawv nqaij hnyav.
Qhov kev sim ob qhov muag tsis pom kev tau ua nyob rau hauv 6 qhov kev sim ua haujlwm hauv lub tebchaws Yelemes. Tag nrho ntawm 404 tus neeg mob uas muaj plaub hau poob tau raug xaiv rau qhov kev sim. Raws li Cassiopeia qhov kev kwv yees, cov kev mob tshwm sim ntawm99% CB-03-01 hmoovyuav tsawg dua li cov tshuaj tiv thaiv androgen hauv khw, xws li finasteride thiab dutasteride.
Khoom Specification
Yam khoom | Specification | Cov txiaj ntsig |
Qhov tshwm sim | Dawb los yog dawb dawb hmoov hmoov | Ua raws |
Kev txheeb xyuas | Los ntawm IR | Ua raws |
Los ntawm HPLC | Ua raws | |
Solubility | Soluble nyob rau hauv DMF, sparingly soluble nyob rau hauv THF, me ntsis soluble nyob rau hauv methanol thiab acetonitrile, heev me ntsis soluble nyob rau hauv ethanol thiab dichloromethane, insoluble nyob rau hauv dej | Ua raws |
Polymorphic Form | Polymorphic daim ntawv 1 | Ua raws |
Melting Point | 211ºC~216ºC | 212.8ºC~214.9ºC |
Cov ntsiab lus dej | Tsawg dua lossis sib npaug rau 0.50% | 0.10% |
Hnyav Hlau | Tsawg dua lossis sib npaug li 10ppm | Ua raws |
Residue ntawm Ignition | Tsawg dua lossis sib npaug rau 0.1% | 0.09% |
Yam khoom | Ib qho impurity: Tsawg dua lossis sib npaug rau 0.1% | 0.03% |
Tag nrho cov impurities: Tsawg dua lossis sib npaug rau 0.9% | 0.15% | |
Assay (ntawm lub hauv paus anhydrous) | 98.0%~102.0% | 99.98% |
Tsis lees paub: tshwj tsis yog tias tau teev tseg, tsab xov xwm kev paub luam tawm los ntawm lub vev xaib no los ntawm Is Taws Nem thiab feem ntau yog siv los txhawb kev sib pauv kev kawm thiab kev kawm. Nws tsis txhais hais tias lub vev xaib no pom zoo nrog nws cov kev xav lossis lees paub qhov tseeb ntawm nws cov ntsiab lus. Thov ua tib zoo tshuaj xyuas nws. Yog tias koj xav tias muaj kev ua txhaum cai hauv tsab xov xwm no, thov hu rau tus thawj tswj hwm. Peb tsis muaj lub luag haujlwm rau qhov tshwm sim ntawm kev siv cov ntaub ntawv thiab kev pabcuam ntawm lub vev xaib no.
Nco tseg: Tag nrho cov tebchaw muaj kev pheej hmoo. Thov nrog koj tus kws qhia ntawv, kws kho mob, lossis lwm tus kws tshawb fawb ua ntej siv. Cov khoom no tsis yog siv los kuaj xyuas, tiv thaiv lossis kho cov kab mob, tab sis tsuas yog siv rau kev tshawb fawb tshawb fawb. Lub tuam txhab tsis muaj lub luag haujlwm rau qhov tshwm sim ntawm kev siv tsis raug.
Yog tias koj xav tau kev pab, thov hu rau peb
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Muaj ntau txoj kev xa khoom rau koj xaiv
Tsheb thauj mus los | Shipping txoj kev | Cargo hnyav xav tau | Qhov zoo |
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7-15 hnub | Los ntawm Cua | Haum rau ntau tshaj 50kg. | |
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