Finasteride yog ib qho inhibitor ntawm 5 reductase -2, uas tsuas tuaj yeem inhibit 5 reductase -2 hauv daim ntawv thov kho mob. Nws yog ib qho enzyme intracellular. Cov mis mos molecular yog C27H3OF6N2O2 thiab qhov hnyav molecular yog 528.5.Avodart hmoovyog hmoov dawb nrog lub melting point ntawm 242 ~ 250 degree, uas yog insoluble nyob rau hauv dej, tab sis soluble nyob rau hauv ethanol (44 mg ml -1), methanol (64 mg ml -1), thiab polyethylene glycol. 400 (3 mg ml-1). Nws yog ib qho tshiab ob zaug inhibitor ntawm 5 reductase, uas tuaj yeem cuam tshuam 5 reductase -1 thiab 5 reductase -2. Piv nrog finasteride, nws tuaj yeem txo DHT concentration (94 .7% vs 70 .8%). Cov nyhuv inhibitory ntawm Avodart ntawm 5 reductase -1 yog 60 npaug ntawm finasteride. 27 lub hlis tom qab noj dutasteride, qhov tshwm sim ntawm prostate cancer yog 50% qis dua li cov placebo pawg.
Nws yog metabolized los ntawm CYP3A4 hauv daim siab. Cov kev sim hauv vitro qhia tau tias CYP3A4 inhibitors xws li ritonavir, ketoconazole, verapamil, diltiazem, cimetidine, thiab ciprofloxacin tuaj yeem ua rau kom cov ntshav siab ntawm cov tazobactam nruab nrab, tab sis tsis muaj kev cuam tshuam pharmacological thiab pharmacokinetic nrog tamsulosin, terazosin, warfarin.
|
|
| Cov duab tiag tiag ntawm Dutasteride hmoov | Dutasteride daim duab kos duab |
Khoom siv
1. Avodart hmoovtuaj yeem siv rau kev kho mob ntawm cov neeg mob benign prostatic hyperplasia.
2. Nws tuaj yeem txhim kho cov tsos mob BPH tau ntev.
3. Nws kuj tuaj yeem txo qhov tshwm sim ntawm tus mob qog noj ntshav prostate.
4. Nws tuaj yeem siv rau prostate o.
5. Nws tuaj yeem siv rau txiv neej alopecia thiab seborrheic alopecia.
6. Nws kuj tuaj yeem siv rau kev kho mob alopecia (cov poj niam thiab menyuam yaus yuav tsum tsis txhob noj).
Khoom Specification
| Yam khoom | Specification | Cov txiaj ntsig |
| Qhov tshwm sim | Dawb los yog yuav luag dawb hmoov | Ua raws |
| Kev txheeb xyuas | Ua tau raws li qhov yuav tsum tau ua | Ua raws |
| Poob rau ziab | Tsawg dua los yog sib npaug rau 0.5% | 0.20% |
| Melting ntau | 246ºC~252ºC | 246ºC~248ºC |
| Cov hlau hnyav | Tsawg dua lossis sib npaug li 20ppm | Ua raws |
| Residue ntawm ignition | Tsawg dua lossis sib npaug rau 0.1% | Ua raws |
| Cov khoom muaj feem xyuam | Loj tshaj Impurities Tsawg dua los yog sib npaug rau 0.5% | 0.33% |
| Tag nrho impurity Tsawg dua lossis sib npaug rau 1.0% | 0.60% | |
| Assay | 98.0%~103.0% | 99.80% |
Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:allen@faithfulbio.comTam sim no.
Koj tuaj yeem tiv tauj kuv ntawm WhatsApp:+86 13137770562





Muaj ntau txoj kev xa khoom rau koj xaiv
Tsheb thauj mus los | Shipping txoj kev | Cargo hnyav xav tau | Qhov zoo |
3-7 hnub | DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD, | Haum rau qis dua 50kg. | Peb muaj warehouses nyob rau hauv lub teb chaws Yelemees thiab California, teb chaws USA, |
7-15 hnub | Los ntawm Cua | Haum rau ntau tshaj 50kg. | |
15-60 hnub | Los ntawm Hiav Txwv | Haum rau ntau tshaj 500kg. |
Tsis lees paub: Cov ntawv luam tawm ntawm lub vev xaib no yog siv los txhawb kev sib pauv kev kawm thiab kev kawm, thiab tsis txhais hais tias lub vev xaib no pom zoo nrog nws cov kev xav lossis lees paub qhov tseeb ntawm nws cov ntsiab lus. Thov lim kom zoo. Yog tias koj ntseeg tias tsab xov xwm no ua txhaum, thov hu rau tus thawj tswj hwm. Peb tsis muaj lub luag haujlwm rau qhov tshwm sim ntawm kev siv cov ntaub ntawv thiab cov kev pabcuam hauv lub vev xaib no.
Nco tseg: Cov tshuaj no yuav tsum tau siv rau kev tshawb fawb nkaus xwb. Cov lus thov no tsis tau raug soj ntsuam los ntawm Food and Drug Administration. Thov nrog koj tus kws kho mob tham thiab kawm txog cov kev tshawb fawb muaj ua ntej siv lawv. Cov khoom no tsis yog tsim los kuaj xyuas, kho, kho lossis tiv thaiv kab mob.
Cim npe nrov: avodart hmoov cas 164656-23-9, lwm tus neeg, manufacturers, hoobkas, lag luam wholesale, yuav, nqe, tej, ntshiab, tsim, kev muag khoom








