Pazopanib hmoov CAS 444731-52-6

Pazopanib hmoov CAS 444731-52-6

Khoom npe: Pazopanib
Synonym: CS-1857
CAS Nr.: 444731-52-6
EINECS NO.:251-228-4
Cov mis mos molecular: C21H23N7O2S
Purity & Qib: 99%; Qib tshuaj
Cim: Dawb hmoov
Cov qauv dawb: Muaj
Tshuag: Hauv Tshuag
Warehouse: USA/EU/AU Warehouse
MOQ & Pob: 10g; Pob raws li xav tau
Shipping: Kev nyab xeeb thiab xa khoom sai
Lub Sijhawm Lead: 7-15 hnub
Khw & Txee lub neej: Txias & qhuav qhov chaw; 24 hli
Xa kev nug
Hauj lwm lawm

 

 
 
Khoom Description
pazopanib powder CAS 444731-52-6
Pazopanib hmoov, muag raws li lub npe nrov Votient, yog tshuaj tiv thaiv kab mob qog noj ntshav thoob ntiaj teb los ntawm Novartis. Nws yog ib qho muaj zog thiab xaiv ntau lub hom phiaj receptor tyrosine kinase inhibitor uas thaiv cov qog loj hlob thiab inhibits angiogenesis. Nws tau raug pom zoo rau lub raum cell carcinoma thiab cov nqaij mos sarcoma los ntawm ntau txoj kev tswj hwm thoob ntiaj teb.Pazopanib yog ntau yam kinase inhibitor uas txwv cov qog loj hlob los ntawm lub hom phiaj angiogenesis ntawm inhibition ntawm enzymes suav nrog vascular endothelial growth factor receptor (VEGFR), platelet-derived growth factor. receptor (PDGFR), c-KIT thiab FGFR.Qhov bioavailability ntawm pazopanib yog 21%, thiab bioavailability ntau ntawm tib neeg yog 14-39%. Cov ntshav siab nce mus txog qhov siab tshaj plaws tom qab qhov nruab nrab ntawm 3.5 teev.
Txoj kev tshawb no muaj txij li 1.0 mus txog 11.9 teev. Thaum siv tsis tu ncua, thaj tsam hauv qab qhov nkhaus (AUC) nce 1.23-4 zaug piv rau ib zaug siv. Kev siv cov tshuaj nrog zaub mov tuaj yeem kwv yees li ob npaug ntawm AUC thiab qhov siab tshaj plaws plasma concentration (Cmax); Crushing ntsiav tshuaj nce AUC los ntawm 1.46 zaug thiab ua ob npaug ntawm Cmax.
Hauv cov ntshav, ntau dua 99.5% ntawm cov khoom raug khi rau plasma proteins. Lub siab enzyme lub luag haujlwm rau cov tshuaj metabolizing yog CYP3A4. CYP1A2 thiab CYP2C8 kuj ua rau me me. Cov metabolites pom nyob rau hauv tib neeg hepatocyte thiab microsomal kuaj muaj xws li ntau yam hydroxyl derivatives thiab tejzaum nws yog carboxylic acid. Tsuas yog 6% ntawm cov khoom siv ncig yog nyob rau hauv daim ntawv ntawm cov metabolites, thiab tag nrho tab sis ib qho ntawm lawv yog 10 mus rau 20 npaug qis dua li pazopanib nws tus kheej. Yog li, cov tshuaj metabolites tsis suav tias yog qhov tseem ceeb rau kev kho mob ntawm cov tshuaj.
pazopanib

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

COA

 

SAIB SPECIFICATION TSEEM CEEB
Qhov tshwm sim Dawb hmoov Ua raws
Physical & ChemicalControl    
Assay >99% 99.18%
tsw Yam ntxwv Ua raws
Poob Thaum Qhuav <0.5% 0.23%
Residue ntawm Ignition Tsawg dua lossis sib npaug rau 1.0% 0.19%
Hnyav Hlau <5ppmMax 0.9ppm
AS <2ppm 0.07ppm
Tshuaj tua kab Tsis zoo Tsis zoo
Microbiological    
Tag Nrho Phaj suav <1000/g Max Ua raws
Poov & Pwm < 100/g Max 18/g
Salmonella Tsis zoo Tsis zoo
E. Coli Tsis zoo Tsis zoo
Xaus Cov khoom no ua raws li cov qauv thoob ntiaj teb

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

Puas yog pazopanib hloov cov plaub hau xim?

Pazopanib yog ib tug multitargeted tyrosine kinase inhibitor siv rau kev kho mob ntawm ntau yam qog malignancies. Cov plaub hau hloov xim, tshwj xeeb tshaj yog cov plaub hau depigmentation, yog ib qho tshwm sim ntawm kev kho pazopanib. Txawm li cas los xij, feem ntau nws maj mam loj hlob dhau ib ntu ntawm ob peb lub hlis.

 

Pazopanib puas tuaj yeem ua rau poob phaus?

mob qhov ncauj los yog rwj, koj lub qhov ncauj kuj yuav qhuav. poob phaus. tsis muaj dej hauv koj lub cev (lub cev qhuav dej) - haus dej kom ntau thaum noj pazopanib. Tam sim ntawd liab ntawm daim tawv nqaij, koj kuj yuav tau txais lwm yam tsos mob xws li tawm hws thiab ib tug sov so.

 

Koj yuav tsum noj dab tsi thaum noj pazopanib?

Tsis txhob noj lossis haus cov txiv kab ntxwv, txiv duaj txiv duaj, txiv kab ntxwv Seville lossis lawv cov kua txiv hmab txiv ntoo (lossis cov khoom uas muaj cov no) thaum kho qhov no. Lawv tuaj yeem ua rau muaj kev phiv ntau ntxiv. Cov tshuaj no tuaj yeem cuam tshuam nrog lwm cov tshuaj thiab tuaj yeem ua rau kev kho mob tsis ua haujlwm zoo lossis ua rau muaj kev phiv loj heev.

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

faithful factory

vim li cas xaiv peb

 
Peb ua raws li lub hauv paus ntsiab lus ntawm "cov neeg siv khoom ua ntej, kev ncaj ncees ua ntej", thiab ib txwm muab cov neeg siv khoom zoo thiab cov khoom siv tau zoo thiab cov kev pabcuam zoo. Xaiv kev ncaj ncees. Xaiv lub neej noj qab nyob zoo!
 
Nrog rau peb cov kev siv zog tas mus li thiab kev pabcuam zoo, peb cia siab tias yuav tsim kev koom tes ntev thiab kev txhim kho nrog cov neeg siv khoom thiab muab sijhawm rau peb. Peb ntseeg tias peb yuav txaus siab rau koj nrog thawj-chav kawm zoo, nyab xeeb thiab xa khoom sai thiab txaus siab rau kev pab cuam tom qab muag.

 

Peb lub Hoobkas

 

faithful-chemical- lab

faithful exhibition

 

Pob

 

faithful-chemical- Packaging

 

Shipping Txoj Kev

 

Tsheb thauj mus los

Shipping txoj kev

Cargo hnyav xav tau

Qhov zoo

3-7 hnub

DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD,
UPS, USPS, FedEx, TNT, EMS

Haum rau qis dua 50kg.
International qhov rooj rau qhov rooj nthuav qhia

Peb muaj warehouses nyob rau hauv lub teb chaws Yelemees thiab California, teb chaws USA, thiab cov neeg muas zaub nyob rau hauv cov teb chaws Europe thiab America muaj peev xwm txaus siab rau xa cov khoom ncaj qha los ntawm ob qhov chaw.

7-15 hnub

Los ntawm Cua

Haum rau ntau tshaj 50kg.
ceev thiab pheej yig dua rau kev txiav txim loj

15-60 hnub

Los ntawm Hiav Txwv

Haum rau ntau tshaj 500kg.
Kev xa khoom pheej yig tshaj plaws

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

Tsis lees paub: Tag nrho cov khoom lag luam (cov khoom siv tsis raug cai) cov duab tau muab coj los ua zoo, tab sis vim yog lub zog ntawm lub teeb (lub sijhawm sib txawv, lub teeb tom qab sib txawv), txoj kev tua, cov khoom siv sib txawv thiab lwm yam, tej zaum yuav muaj qee qhov sib txawv ntawm qhov daim duab thiab cov xim tiag tiag, cov khoom xim, thov coj cov nyhuv tiag tiag, cov khoom xim sib txawv tsis yog qhov teeb meem ntawm cov khoom zoo.
 
Nco tseg: Nco ntsoov sab laj nrog tus kws kho mob uas tsim nyog ua ntej noj cov tshuaj tshiab. Cov khoom no tsis yog tsim los kuaj xyuas, kho, kho lossis tiv thaiv txhua yam kab mob.Thaum lub sijhawm yuav khoom, tus neeg yuav khoom thoob ntiaj teb pom zoo xav tias muaj kev pheej hmoo ntawm txhua yam khoom tuaj txog. Peb tsis tuaj yeem hloov cov khoom ploj lossis raug kaw. Ua ntej xa cov khoom, koj yuav tsum paub meej tias koj pom zoo rau cov nqe lus no.Qhov no tsuas yog kev pom zoo koob tshuaj raws li peb tus kheej cov kev paub dhau los thiab cov ntaub ntawv pov thawj. Peb pom zoo kom koj ua koj tus kheej kev tshawb fawb ua ntej siv cov khoom no.

 

Cim npe nrov: pazopanib hmoov cas 444731-52-6, Suav teb, lwm tus neeg, manufacturers, hoobkas, customized, lag luam wholesale, yuav, nqe, tej, ntshiab, tsim, luv nqi, muag, Tshuag, dawb qauv, raw hmoov, raw khoom, ua nyob rau hauv Tuam Tshoj