Sitagliptin hmoov CAS 486460-32-6

Sitagliptin hmoov CAS 486460-32-6

Khoom npe: Sitagliptin
Synonym: Sitagliptin puag; Sitagliptin-D4; Sitagliptin-D4 HCL; Janumet
CAS Nr.: 486460-32-6
EINECS NO.:690-730-1
Cov roj formula: C16H15F6N5O
Purity & Qib: 99%; Qib tshuaj
Cim: Dawb hmoov
Cov qauv dawb: Muaj
Tshuag: Hauv Tshuag
Warehouse: USA/EU/AU Warehouse
MOQ & Pob: 1g; Pob raws li xav tau
Shipping: Kev nyab xeeb thiab xa khoom sai
Lub Sijhawm Lead: 7-15 hnub
Khw & Txee lub neej: Txias & qhuav qhov chaw; 24 hli
Xa kev nug
Hauj lwm lawm

 

 
 
Khoom Description
Sitagliptin effect
Sitagliptin, ib yam tshiab ntawm cov tshuaj tiv thaiv kab mob ntshav qab zib hom II, yog thawj dipeptidyl peptidase -Ⅳ (DPP-Ⅳ) inhibitor siv los kho mob ntshav qab zib hom II, uas feem ntau siv los ua phosphate. Sitagliptin tuaj yeem tiv thaiv thiab kho mob ntshav qab zib hom 2, hyperglycemia, insulin tsis kam, rog, ntshav siab thiab qee yam teeb meem.
 
Cov txheej txheem ntawm sitagliptin txawv ntawm cov neeg ua haujlwm hypoglycemic yav dhau los. Nws tuaj yeem tswj hwm cov ntshav qab zib ntawm cov neeg mob ntshav qab zib los ntawm kev txhim kho lub peev xwm ntawm islet cells los tsim cov tshuaj insulin thiab ua kom cov tshuaj insulin tso tawm thaum cov ntshav qab zib nce.
Sitagliptin yog tshuaj rau cov neeg uas tseem muaj ntshav qab zib ntau, txawm tias lawv muaj kev noj qab haus huv thiab kev tawm dag zog tsis tu ncua. Nws ua haujlwm los ntawm kev nce cov tshuaj insulin uas koj lub cev ua. Insulin yog cov tshuaj hormones uas tswj cov piam thaj hauv koj cov ntshav.
 
Sigliptin, nrog lub npe lag luam Jiatangwei, yog tus neeg sawv cev hypoglycemic (antidiabetic tus neeg sawv cev) thiab belongs rau dipeptidyl peptidase -4(DPP-4) inhibitor. Siglitazone tuaj yeem siv ib leeg lossis ua ke nrog lwm cov tshuaj hypoglycemic los kho cov ntshav qab zib hom 2 (xws li metformin lossis thiazolidinedione). Qhov kom zoo dua ntawm sitagliptin yog tias muaj kev phiv tsawg dua (xws li txo qis ntawm hypoglycemia thiab qhov hnyav nce) thaum tswj cov piam thaj hauv cov ntshav. Txawm hais tias kev nyab xeeb yog nws qhov zoo dua, nws cov nyhuv tsis tuaj yeem lav tau zoo, yog li nws feem ntau pom zoo kom ua ke nrog lwm yam tshuaj xws li metformin.
Sitagliptin analysis

 

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COA

 

Yam khoom Specification Cov qhabnias xeem
Yam ntxwv Dawb hmoov Ua raws
Assay Ntau dua lossis sib npaug rau 99.0% 99.15%
Poob rau ziab Tsawg dua lossis sib npaug rau 2.0% 1.65%
Pb Tsawg dua lossis sib npaug rau 2.0PPM Ua raws
Raws li Tsawg dua lossis sib npaug rau 1.0PPM Ua raws
Hg Tsawg dua lossis sib npaug rau 0.5PPM Ua raws
Tag Nrho Phaj suav Tsawg dua lossis sib npaug li 1000CFU / g Ua raws
Poov / Pwm Tsawg dua lossis sib npaug li 100CFU / g Ua raws
E. Coli Tsis zoo Ua raws
Xaus Ua raws li kev lag luam specification

 

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Yam khoom

 

  • Qhov ceev 1.6 ± 0.1g / cm3

  • Kub taw tes 529.9 ± 6 0.0 degree ntawm 760 mmHg

  • Cov mis mos molecular C16H15F6N5O

  • Molecular hnyav 407.314

  • Flash point 274.3 ± 32.9 degree

  • Qhov tseeb loj 407.118073

Sitagliptin MF

 

Yam tshuaj twg yog sitagliptin?

Sitagliptin yog nyob rau hauv ib chav kawm ntawm cov tshuaj hu ua dipeptidyl peptidase -4 (DPP-4) inhibitors. Nws ua hauj lwm los ntawm kev nce cov nqi ntawm tej yam ntuj tso uas txo cov ntshav qab zib thaum nws siab.

 

Puas yog sitagliptin yog GLP-1?

Sitagliptin yog ib tug tswv cuab ntawm cov chav kawm gliptin ntawm cov tshuaj tiv thaiv kab mob. Nws cov txheej txheem ntawm kev ua haujlwm yog los ntawm inhibition ntawm dipeptidyl peptidase-4 (DPP-4), ib qho enzyme uas ua rau degrade thiab inactivate glucagon-zoo li peptide-1 (GLP-1).

 

Puas yog sitagliptin thiab metformin tib yam?

Metformin txo qhov nqus ntawm cov piam thaj los ntawm lub plab, txo qis cov piam thaj hauv lub siab, thiab pab koj lub cev siv cov suab thaj zoo dua. Sitagliptin pab tswj cov ntshav qab zib ntau ntxiv los ntawm kev nce cov tshuaj hauv lub cev uas ua rau cov txiav tso tawm insulin ntau dua.

 

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faithful factory

vim li cas xaiv peb

 
Peb ua raws li lub hauv paus ntsiab lus ntawm "cov neeg siv khoom ua ntej, kev ncaj ncees ua ntej", thiab ib txwm muab cov neeg siv khoom zoo thiab cov khoom siv tau zoo thiab cov kev pabcuam zoo. Xaiv kev ncaj ncees. Xaiv lub neej noj qab nyob zoo!
 
Nrog rau peb cov kev siv zog tas mus li thiab kev pabcuam zoo, peb cia siab tias yuav tsim kev koom tes ntev thiab kev txhim kho nrog cov neeg siv khoom thiab muab sijhawm rau peb. Peb ntseeg tias peb yuav txaus siab rau koj nrog thawj-chav kawm zoo, nyab xeeb thiab xa khoom sai thiab txaus siab rau kev pab cuam tom qab muag.

 

Peb lub Hoobkas

 

faithful-chemical- lab

faithful exhibition

 

Pob

 

faithful-chemical- Packaging

 

Shipping Txoj Kev

 

Tsheb thauj mus los

Shipping txoj kev

Cargo hnyav xav tau

Qhov zoo

3-7 hnub

DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD,
UPS, USPS, FedEx, TNT, EMS

Haum rau qis dua 50kg.
International qhov rooj rau qhov rooj nthuav qhia

Peb muaj warehouses nyob rau hauv lub teb chaws Yelemees thiab California, teb chaws USA, thiab cov neeg muas zaub nyob rau hauv cov teb chaws Europe thiab America muaj peev xwm txaus siab rau xa cov khoom ncaj qha los ntawm ob qhov chaw.

7-15 hnub

Los ntawm Cua

Haum rau ntau tshaj 50kg.
ceev thiab pheej yig dua rau kev txiav txim loj

15-60 hnub

Los ntawm Hiav Txwv

Haum rau ntau tshaj 500kg.
Kev xa khoom pheej yig tshaj plaws

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

Tsis lees paub: Tag nrho cov khoom lag luam (cov khoom siv tsis raug cai) cov duab tau muab coj los ua zoo, tab sis vim yog lub zog ntawm lub teeb (lub sijhawm sib txawv, lub teeb tom qab sib txawv), txoj kev tua, cov khoom siv sib txawv thiab lwm yam, tej zaum yuav muaj qee qhov sib txawv ntawm qhov daim duab thiab cov xim tiag tiag, cov khoom xim, thov coj cov nyhuv tiag tiag, cov khoom xim sib txawv tsis yog qhov teeb meem ntawm cov khoom zoo.
 
Nco tseg: Nco ntsoov sab laj nrog tus kws kho mob uas tsim nyog ua ntej noj cov tshuaj tshiab. Cov khoom no tsis yog tsim los kuaj xyuas, kho, kho lossis tiv thaiv txhua yam kab mob.Thaum lub sijhawm yuav khoom, tus neeg yuav khoom thoob ntiaj teb pom zoo xav tias muaj kev pheej hmoo ntawm txhua yam khoom tuaj txog. Peb tsis tuaj yeem hloov cov khoom ploj lossis raug kaw. Ua ntej xa cov khoom, koj yuav tsum paub meej tias koj pom zoo rau cov nqe lus no.Qhov no tsuas yog kev pom zoo koob tshuaj raws li peb tus kheej cov kev paub dhau los thiab cov ntaub ntawv pov thawj. Peb pom zoo kom koj ua koj tus kheej kev tshawb fawb ua ntej siv cov khoom no.

 

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