Tacrolimus hmoov CAS 104987-11-3
Khoom npe: Tacrolimus
Lub ntsiab lus: Advagraf; Protopic; Tacrolimus; Suniti; Prograf
CAS Nr.: 104987-11-3
EINECS NO.:1308068-626-2
Cov roj formula: C44H69NO12
Purity & Qib: 99%; Qib tshuaj
Cim: Dawb hmoov
Cov qauv dawb: Muaj
Tshuag: Hauv Tshuag
Warehouse: USA/EU/AU Warehouse
MOQ & Pob: 1g; Pob raws li xav tau
Shipping: Kev nyab xeeb thiab xa khoom sai
Lub Sijhawm Lead: 7-15 hnub
Khw & Txee lub neej: Txias & qhuav qhov chaw; 24 hli
Hauj lwm lawm
Khoom piav qhia

Tachlimusyog ib hom tshuaj macrolide cais tawm ntawm Streptomyces. Nws muaj lub zog tiv thaiv kab mob, uas muaj peev xwm tshwj xeeb khi rau thiab inhibit calmodulin phosphatase kev ua, inhibit IL-2 signaling transcription, thiab yog li inhibit T cell activation, TNF-, IL-1 thiab IL{{4} } ntau lawm, thiab T-cell-dependent B cell proliferation. Piv nrog rau cyclosporine, lwm tus calmodulin phosphatase inhibitor, tacrolimus inhibited T cell ua kom muaj zog ntau dua nrog cov teebmeem tsis zoo.
Tacrolimus (tseem hu ua FK506, lub npe lag luam: Precofu), tau siv dav hauv ntau yam kev hloov pauv hauv nruab nrog cev tom qab kev tiv thaiv kev tsis lees paub, tab sis kuj siv los kho cov kab mob autoimmune, kab mob raum, kab mob hauv cov ntshav.
Txawm li cas los xij, kev siv tacrolimus sib txawv ntawm cov tib neeg, thiab ntau yam tshuaj thiab khoom noj tuaj yeem cuam tshuam rau qib tacrolimus ntawm txhua theem ntawm kev siv.
Tacrolimusyog tshuaj tua kab mob macrolide. Cov tshuaj tiv thaiv kab mob. Cov txheej txheem ntawm kev ua yog tib yam li ntawm cyclosporin, feem ntau inhibiting cov synthesis ntawm interleukin -2. Nws yog siv rau kev hloov pauv hauv nruab nrog cev tsis lees paub thiab muaj txiaj ntsig zoo dua rau kev tsis lees paub.
McNeill thiab Koo tau hais tias tsiaj thiab tib neeg cov kev tshawb fawb qhia tias cov tshuaj pleev tacrolimus yog ib qho kev nyab xeeb rau cov tshuaj steroids, nrog rau kev kub hnyiab nkaus xwb raws li qhov paub txog qhov tsis zoo piv nrog cov tshuaj steroids, nrog rau cov kev mob tshwm sim ntev.

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COA
Kev sim | Specification | Cov txiaj ntsig |
Qhov tshwm sim | Dawb los yog yuav luag dawb crystalline hmoov | Ua raws |
Kev txheeb xyuas | IR | Ua raws |
HPLC | Ua raws | |
Dej | 1.6% rau 3.0%Max | 2.30% |
Residue ntawm lgnition | 0.2% Max | 0.01% |
Hnyav Hlau | 20 PPM Max | Ua raws |
Yam khoom muaj feem | Ascomycin 0.8% Max | 0.05% |
Dihydrotacrolimus 0.6% Max | 0.30% | |
Tag nrho impurities 1.5% Max | 0.43% | |
Residual Solvents | Acetone 2000PPM Max | Tsis Pom |
Ethanol 2000PPM Max | Tsis Pom | |
Assay (lub hauv paus qhuav) | 98% mus rau 102% | 99.00% |
Xaus | Mus txog Standard rau Export |
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Cov tshuaj tacrolimus siv rau dab tsi?
Tacrolimus yog siv ua ke nrog lwm cov tshuaj los tiv thaiv lub cev los ntawm kev tsis lees txais ib qho kev hloov pauv hauv nruab nrog cev (xws li lub raum, siab, lub plawv, lossis lub ntsws). Cov tshuaj no tuaj yeem siv nrog steroids, azathioprine, basiliximab, lossis mycophenolate mofetil. Tacrolimus belongs rau ib pawg tshuaj hu ua immunosuppressive agents.
Puas yog tacrolimus yog cov tshuaj uas pheej hmoo siab?
Tacrolimus yog tshuaj muaj zog heev. Nws tuaj yeem ua rau muaj kev phiv loj heev, xws li teeb meem raum. Nws kuj tseem tuaj yeem txo lub cev muaj peev xwm tiv thaiv kab mob. Koj thiab koj tus kws kho mob yuav tsum tham txog cov txiaj ntsig ntawm cov tshuaj no nrog rau kev pheej hmoo ntawm kev siv nws.
Puas yog tacrolimus yog tshuaj khomob?
Tacrolimus yog nyob rau hauv ib chav kawm ntawm cov tshuaj hu ua immunosuppressants. Nws ua haujlwm los ntawm kev txo qis kev ua haujlwm ntawm lub cev tiv thaiv kab mob los tiv thaiv nws los ntawm kev tawm tsam cov kabmob hloov pauv.
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Pob
Shipping Txoj Kev
Tsheb thauj mus los |
Shipping txoj kev |
Cargo hnyav xav tau |
Qhov zoo |
3-7 hnub |
DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD, |
Haum rau qis dua 50kg. |
Peb muaj warehouses nyob rau hauv lub teb chaws Yelemees thiab California, teb chaws USA, thiab cov neeg muas zaub nyob rau hauv cov teb chaws Europe thiab America yuav txaus siab rau xa cov khoom ncaj qha los ntawm ob qhov chaw. |
7-15 hnub |
Los ntawm Cua |
Haum rau ntau tshaj 50kg. |
|
15-60 hnub |
Los ntawm Hiav Txwv |
Haum rau ntau tshaj 500kg. |
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