Varenicline Tartrate yog dab tsi?
Varenicline Tartrate yog ib feem agonist ntawm 4 2 nAChR nicotinic acetylcholine receptor (EC50=2.3 μM). Varenicline Tartrate yog ib tug ua tiav agonist ntawm 3 4 nAChR thiab 7 nAChR acetylcholine receptors nrog EC50 qhov tseem ceeb ntawm 55 μM thiab 18 μM, feem. Varenicline yog ib qho nicotine ligand raws li cov qauv cytosine, uas tuaj yeem txo cov nicotine craving thiab tshem tawm cov tsos mob, thiab tuaj yeem pab txo kev haus luam yeeb hauv 12 lub lis piam ntawm kev kho mob.
Varenicline tartrate yog cov organic compound, thiabVarenicline tartrate hmoovyog xim tsis muaj xim lossis crystalline hmoov nrog cov txiv hmab txiv ntoo qaub saj.

| Khoom npe | Varenicline Tartrate |
| CAS | 375815-87-5 |
| Cov mis mos molecular | C17H19N3O6 |
| Molecular hnyav | 361.35 |
| EINECS Number | 638-780-5 |
| Kev cia khoom | chav kub |
| Melting point | 206-208 degree |
| Solubility | Dimethyl sulfoxide:> 5mg / mL |
| Qhov tshwm sim | Dawb hmoov |
| Boiling point | 400.6 degree ntawm 760 mmHg |
| MOQ |
100g |
Varenicline tartrate ua haujlwm li cas?
Tom qabVarenicline tartrate hmoovkhi rau nicotinic acetylcholine receptor, ntawm ib sab, nws ua raws li agonist los txhawb kev tso tawm ntawm dopamine hauv lub hlwb, uas tuaj yeem txo cov tsos mob tshem tawm tom qab txiav luam yeeb; Ntawm qhov tod tes, nws cov khoom antagonistic tuaj yeem tiv thaiv nicotine los ntawm kev sib txuas nrog nicotine acetylcholine receptor thiab txo qhov kev zoo siab ntawm kev haus luam yeeb.
Khoom Specification
| Yam khoom | Specification | Cov txiaj ntsig |
| Qhov tshwm sim | Dawb hmoov | Ua raws |
| Kev txheeb xyuas | Los ntawm HPLC | Ua raws |
| Melting Point | 206-208 degree | Ua raws |
| Poob rau ziab | Tsawg dua lossis sib npaug rau 1.00% | 0.21% |
| Hnyav Hlau | Tsawg dua lossis sib npaug li 10ppm | Ua raws |
| Sulfated tshauv | Tsawg dua lossis sib npaug rau 0.10% | 0.03% |
| Cov ntsiab lus | 17.5%~19.5% | 19.3% |
| Cov ntsiab lus | Tsawg dua lossis sib npaug rau 0.1ppm | 0.09ppm |
| Ua VContent | Tsawg dua los yog sib npaug rau 3.0ppm | 0.50ppm |
| Cov ntsiab lus | Tsawg dua lossis sib npaug rau 0.1ppm | 0.10ppm |
| Cov ntsiab lus | Tsawg dua lossis sib npaug rau 0.1ppm | 0.10ppm |
| Microbiological Test | Coliforms: Tsis zoo | Tsis zoo |
| Salmonella: Tsis zoo | Ua raws | |
| Tag nrho cov phaj suav: Tsawg dua lossis sib npaug rau 1000 CFU / g | Hla | |
| Poov xab & Pwm: Tsawg dua lossis sib npaug li 50 CFU / g | Hla | |
| Yam khoom muaj feem | Impurity A: Tsawg dua lossis sib npaug rau 0.30% | 0.18% |
| Lwm yam impurity tsis paub: Tsawg dua lossis sib npaug rau 0.10% | 0.07% | |
| Tag nrho cov impurities: Tsawg dua lossis sib npaug rau 0.50% | 0.42% | |
| Assay | Ntau dua lossis sib npaug rau 99.0% | 99.5% |
| Daim ntawv pov thawj | USP Txuj | |
| Xaus | Cov khoom ua tau raws li USP tus qauv. | |
Dab tsi yog qhov cuam tshuam ntawm Varenicline tartrate?
1. Tswj kev haus luam yeeb:Varenicline Tartrate hmoovtuaj yeem inhibit qhov nqus ntawm nicotine thiab txo qhov kev xav tau ntawm kev haus luam yeeb los ntawm kev tswj hwm qib dopamine. Yog li ntawd, nws tuaj yeem tswj tau kev haus luam yeeb zoo thiab pab cov neeg mob txiav luam yeeb.
2. Txhim kho txoj kev ua pa: Vim muaj cov tshuaj tiv thaiv kab mob ntawm Varenicline Tartrate, nws tuaj yeem pab txhim kho kev ua pa ntawm cov neeg mob, yog li txo cov tsos mob xws li hnoos thiab ua tsis taus pa ntsig txog kev haus luam yeeb.
3. Txo kev ntxhov siab: Kev haus luam yeeb ntev ntev yuav ua rau muaj kev ntxhov siab thiab lwm yam teeb meem puas siab ntsws. Cov kev tshawb fawb tau pom tias Varenicline Tartrate tuaj yeem txo cov tsos mob no los ntawm kev tswj cov qib dopamine.
4. Txhawb kev pw tsaug zog zoo: Kev haus luam yeeb yuav cuam tshuam rau kev pw tsaug zog zoo. Kev tshawb fawb qhia tau tias Varenicline Tartrate muaj txiaj ntsig los txhim kho kev pw tsaug zog zoo thiab ua kom lub sijhawm pw tsaug zog ntev.
HTML5 atlas ntawm Varenicline tartrate
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Dab tsi yog kev ceev faj ntawm Varenicline tartrate?
1, yuav tsum tau siv tshuaj raws li kev qhia ntawm tus kws kho mob;
2, tsis tuaj yeem nres noj tshuaj lossis hloov cov koob tshuaj tam sim ntawd;
3, ua ke nrog lwm cov tshuaj sedatives thiab central paj hlwb depressants yuav tsum ceev faj;
4. Nws muaj kev cuam tshuam rau cawv thiab lwm yam tshuaj tiv thaiv.
Yuav ua li cas thiab qhov twg yuav Varenicline Tartrate Powder wholesale?
Koj tuaj yeem tso siab rau peb qhov kev txiav txim vim tias peb muaj cov ntaub ntawv zoo ntawm kev muag tshuaj raws cai.
Peb ua qhov kev kuaj xyuas ywj pheej ntawm txhua yam khoom thiab tom qab ntawd muag rau peb cov neeg siv khoom hwm.
Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:allen@faithfulbio.comTam sim no.





Muaj ntau txoj kev xa khoom rau koj xaiv
|
Tsheb thauj mus los |
Shipping txoj kev |
Cargo hnyav xav tau |
Qhov zoo |
|
3-7 hnub |
DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD, |
Haum rau qis dua 50kg. |
Peb muaj warehouses nyob rau hauv lub teb chaws Yelemees thiab California, teb chaws USA, |
|
7-15 hnub |
Los ntawm Cua |
Haum rau ntau tshaj 50kg. |
|
|
15-60 hnub |
Los ntawm Hiav Txwv |
Haum rau ntau tshaj 500kg. |
Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:allen@faithfulbio.comTam sim no.
Tsis lees paub: Cov ntawv luam tawm ntawm lub xaib no yog siv los txhawb kev sib pauv kev kawm thiab kev kawm, thiab tsis txhais hais tias lub vev xaib no pom zoo nrog nws cov kev xav lossis lees paub qhov tseeb ntawm nws cov ntsiab lus. Thov lim kom zoo. Yog tias koj ntseeg tias tsab xov xwm no ua txhaum, thov hu rau tus thawj tswj hwm. Peb tsis muaj lub luag haujlwm rau qhov tshwm sim ntawm kev siv cov ntaub ntawv thiab cov kev pabcuam hauv lub vev xaib no.
Nco tseg: Cov tshuaj no yuav tsum tau siv rau kev tshawb fawb nkaus xwb. Cov lus thov no tsis tau raug soj ntsuam los ntawm Food and Drug Administration. Thov nrog koj tus kws kho mob tham thiab kawm txog cov kev tshawb fawb muaj ua ntej siv lawv. Cov khoom no tsis yog tsim los kuaj xyuas, kho, kho, lossis tiv thaiv txhua yam kab mob.
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