J 147 Hmoov CAS 1146963-51-0

J 147 Hmoov CAS 1146963-51-0

Khoom npe: J 147 hmoov
CAS TSIS MUAJ .: 90038-01-0
Molecular cov mis: c18h17f3n2o2
Einec.No:1592732-453-0
Txhais tau: J 147; J-147; CS-1446
Shipping: DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD, UPS, USPS, EMS, los ntawm huab cua, los ntawm hiav txwv thiab lwm yam
Khw & txee lub neej: txias & qhov chaw qhuav; 36 lub hlis
Lwm yam: Muaj cov chaw khaws khoom hauv Tebchaws Meskas, Australia thiab Yelemes
Xa kev nug
Hauj lwm lawm

Dab tsi yog J 147 hmoov?

J 147 hmoovyog ib tus neeg saib xyuas muaj txiaj ntsig zoo rau cov neeg saib xyuas uas muaj peev xwm ua kom muaj peev xwm txhim kho kev txawj ntse. J - 147 tuaj yeem dhau los ntawm cov ntshav lub hlwb (BBB). J-147 inhibits monoamine oxidase b (maob) thiab dopamine transporter, nrog EC50 tseem ceeb ntawm 1.88 μ m, ntsig txog. J-147 muaj peev xwm rau kev tshawb fawb txog Alzheimer tus kab mob (ad).

MF of J 147 powder CAS 1146963-51-0

Khoom npe

J 147

Cas

1146963-51-0

Molecular Cov Qauv

C18H17F3N2O2
Einecs 1592732-453-0

Molecular hnyav

350.33
Kub taw tes 412.8 ± 55.0 Degree (kwv yees)

Kev tshwm sim

Cov hmoov dawb

Ceev 1.18 ± 0.1 g / cm3 (kwv yees)

 

Dab tsi yog qhov tseem ceeb ntawm J 147 hmoov?

J 147 muaj cov hom phiaj hauv qab no

  • Alzheimer Kev Tshawb Fawb Txog Kab Mob

J 147 yog ntau - Lub Hom Phiaj Me Me Me Kev Tshawb Fawb, thiab J-147 Kev Tshawb Fawb Cov Khoom Siv Alzheimer, thiab Kev Ntsuam Xyuas Yeeb Tshuaj, thiab muaj peev xwm kho cov kab mob.

  • Neuroprotective effect

Cov kev sim tau pom tias nws yuav tiv thaiv cov neurons los ntawm kev tiv thaiv neuroinofammegation, thiab txhim kho mitochondrial muaj nuj nqi. Cov hmoov qub qub tuaj yeem siv tau rau cov kev sim ua lag luam pharcacological.

J147 can improve memory ability

  • Kev Tsim Kho Yeeb Tshuaj thiab Kev Txhim Kho

Raws li cov khoom siv nquag ntawm cov tshuaj sib tw, cov hmoov nplej nyoos tuaj yeem txhawb kev tshawb fawb theem xws li kev txheeb xyuas cov tshuaj (PK / PD), kev sib tw toxicity.

  • Kev sib piv thiab cov qauv khoom lag luam
Hauv chav kuaj, J 147 siv tau los ua kev tswj hwm zoo lossis qauv los piv cov kev ua si ntawm lwm cov chaw sib txuas lossis txheeb xyuas qhov tseeb ntawm cov qauv sim.
  • Kev tshawb fawb txog kev cuam tshuam synergistic
Nws tuaj yeem siv ua ke nrog lwm cov tshuaj lossis cov khoom lag luam los tshawb txog kev kho mob lossis nthuav dav nws xav tau, pls nyem e {}}}}sales1@faithfulbio.com

Khoom Qhia Txog Khoom

Cov khoom Kev qhia tshwj xeeb Qho kawg
Kev tshwm sim Dawb rau tawm - Cov hmoov nplej dawb Ua raws
Daim qhia npe Ob NMR thiab MS cov ntaub ntawv yeej muaj raws li cov lus qhia hauv cov ntawv Ua raws
So Soluble hauv dmo Ua raws
Assisy (ntawm lub anhydrous hauv paus) 98.0%~102.0% 99.3%
Xaus:Ua raws li kev lag luam tshwj xeeb

 

J 147 hmoov ua haujlwm li cas?

Mechanism of J 147

J 147 hmoovUa raws li neuroprotrophic thiab neurotrophic compound los ntawm inhibiting atp5a, tus tseem ceeb enzyme nyob rau hauv kev laus. Nws kuj tseem zoo li txhim kho kev tsim cov hlwb - derived neurotrophic factor (BDNF), uas pab neurons.

Qhov cuam tshuam hauv tsiaj qauv:

Tiv thaiv cov neurotoxicity hauv cov xovtooj ntawm tes.

Txo cov qib amyloid - beta peptides thiab nce BDNF hauv cov hippocampus ntawm nas.

Txhim kho cov nas.

Tiv thaiv kev nco tsis nco qab hauv Alzheimer's - qauv mice.

Qhia txog cov peev xwm rau lwm yam xwm txheej zoo li kev raug mob lub hlwb.

 

Yuav ua li cas los tsim J 147 hmoov?

how to produce J147

 

Maj mam ntxiv trifluoroacetic anhydride herdride (0.33ml, 2.36g, 1.97mmide (0.33ml, 2.36mm) hauv dichhlorometomethane (5ml) ntawm 0℃thiab nyob rau hauv nitrogen tiv thaiv. Cov tshuaj tiv thaiv sib xyaw tau raug ntsia tsis tu ncua ntawm 0℃rau 1.5 teev. Tom qab cov tshuaj tiv thaiv tau ua tiav, cov sib xyaw kom muaj zog, thiab cov seem yog huv si los ntawm kem chromatography siv a (1:10) sib xyaw ua ke raws li cov khoom lag luamJ 147 hmoov(571 mg, tawm los 83%).

 

Yuav ua li cas thiab qhov twg yuav J 147 hmoov?

Peb muaj 8 xyoo kev paub hauv kev muag cov tshuaj tshawb fawb txog kev cai lij choj thiab muaj lub koob npe zoo, ua rau peb tus khub uas ntseeg siab.
Peb paub tseeb tias qhov zoo ntawm peb cov khoom los ntawm kev sim ua haujlwm ywj pheej, thiab txhua tus neeg siv khoom yog peb VIP.

Xa koj qhov kev nug kom paub ntau ntxiv, Nyem Email:sales1@faithfulbio.comTam sim no.

 

J 147 powder

J 147 powder

J 147 powder

J 147 powder

J 147 powder

 

Ntau hom kev xa khoom rau koj xaiv

Tsheb Thauj Mus Los

Shipping Txoj Kev

Cargo Qhov hnyav

Yam uas pab

3-7 hnub

DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD,
UPS, USPS, FedEx, TNT, EMS

Haum rau hauv qab 50kg.
Lub qhov rooj thoob ntiaj teb rau qhov rooj Express

Peb muaj cov chaw khaws khoom hauv Tebchaws Yelemees thiab California, Asmeskas,
thiab cov neeg muas zaub hauv Tebchaws Europe thiab Asmeskas tau
Txaus siab rau xa cov khoom ncaj qha los ntawm ob qhov chaw no.

7-15 hnub

Los ntawm huab cua

Haum rau ntau tshaj 50kg.
nrawm thiab pheej yig dua rau kev txiav txim loj

15-60 hnub

Los ntawm hiav txwv

Haum rau ntau tshaj 500kg.
Pheej Yig Tshaj Qho Kev Lag Luam

Cov FAQ

Q: Puas muaj kev phiv los ntawm J 147?

A: Lub siab bioavailability thiab ntshav - cov nyhuv rau nws cov kev cuam tshuam lub hlwb, tsis muaj ib qho tseem ceeb ntawm J147 tau tshaj tawm.

Q: Lub neej ntawm J 147 hmoov dab tsi?

A: (E / Z) - j147 ntsig txog cov tshuaj tiv thaiv kab mob
Ib nrab lub neej (t1/2) Ntawm (E / Z) {- J147 tau muab xam thaum 1.5 hrs hauv 1.5 teev hauv lub hlwb (PO) kev tswj hwm ntawm ib koob ntawm 20 mg / kg).

Q: J 147 nrhiav tau li cas?

A: J147 tau tsim kho xyoo 2011. J147 yog hloov kho version ntawm cov molecule (curcumin) pom nyob rau hauv curry Spice Turmeric.

 

Kev tsis lees paub: Cov lus ntawm lub vev xaib no yog siv rau kev tshawb fawb thiab kev kawm sib pauv. Thov ua tib zoo saib pom qhov tseeb ntawm lawv cov kev xav thiab cov ntsiab lus. Yog tias koj pom muaj kev ua txhaum. Thov hu rau tus thawj tswj hwm kom sai. Peb tsis yog lub luag haujlwm rau cov kev rau txim ntawm cov ntaub ntawv thiab cov kev pabcuam tau muab rau hauv lub vev xaib no.

 

Tsab ntawv: Cov khoom lag luam yog rau kev tshawb fawb tsuas yog siv thiab tsis yog rau kev kuaj mob, kev kho mob, tiv thaiv kab mob, thiab lwm yam.

 

Xa koj qhov kev nug kom paub meej ntxiv, nyem email:sales1@faithfulbio.comTam sim no.

 

Cim npe nrov: J 147 Hmoov CAS 1146963-51-0, Tuam Tshoj Tuam Tshoj, Cov Qauv, Kev Muag Khoom, Khoom Siv Dawb, Khoom Siv Raw, Ua Hauv Suav