Dab tsi yog J 147 hmoov?
J 147 hmoovyog ib tus neeg saib xyuas muaj txiaj ntsig zoo rau cov neeg saib xyuas uas muaj peev xwm ua kom muaj peev xwm txhim kho kev txawj ntse. J - 147 tuaj yeem dhau los ntawm cov ntshav lub hlwb (BBB). J-147 inhibits monoamine oxidase b (maob) thiab dopamine transporter, nrog EC50 tseem ceeb ntawm 1.88 μ m, ntsig txog. J-147 muaj peev xwm rau kev tshawb fawb txog Alzheimer tus kab mob (ad).
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Khoom npe |
J 147 |
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Cas |
1146963-51-0 |
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Molecular Cov Qauv |
C18H17F3N2O2 | |
| Einecs | 1592732-453-0 | |
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Molecular hnyav |
350.33 | |
| Kub taw tes | 412.8 ± 55.0 Degree (kwv yees) | |
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Kev tshwm sim |
Cov hmoov dawb |
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| Ceev | 1.18 ± 0.1 g / cm3 (kwv yees) |
Dab tsi yog qhov tseem ceeb ntawm J 147 hmoov?
J 147 muaj cov hom phiaj hauv qab no
- Alzheimer Kev Tshawb Fawb Txog Kab Mob
J 147 yog ntau - Lub Hom Phiaj Me Me Me Kev Tshawb Fawb, thiab J-147 Kev Tshawb Fawb Cov Khoom Siv Alzheimer, thiab Kev Ntsuam Xyuas Yeeb Tshuaj, thiab muaj peev xwm kho cov kab mob.
- Neuroprotective effect
Cov kev sim tau pom tias nws yuav tiv thaiv cov neurons los ntawm kev tiv thaiv neuroinofammegation, thiab txhim kho mitochondrial muaj nuj nqi. Cov hmoov qub qub tuaj yeem siv tau rau cov kev sim ua lag luam pharcacological.
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Raws li cov khoom siv nquag ntawm cov tshuaj sib tw, cov hmoov nplej nyoos tuaj yeem txhawb kev tshawb fawb theem xws li kev txheeb xyuas cov tshuaj (PK / PD), kev sib tw toxicity.
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Khoom Qhia Txog Khoom
| Cov khoom | Kev qhia tshwj xeeb | Qho kawg |
| Kev tshwm sim | Dawb rau tawm - Cov hmoov nplej dawb | Ua raws |
| Daim qhia npe | Ob NMR thiab MS cov ntaub ntawv yeej muaj raws li cov lus qhia hauv cov ntawv | Ua raws |
| So | Soluble hauv dmo | Ua raws |
| Assisy (ntawm lub anhydrous hauv paus) | 98.0%~102.0% | 99.3% |
| Xaus:Ua raws li kev lag luam tshwj xeeb | ||
J 147 hmoov ua haujlwm li cas?
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J 147 hmoovUa raws li neuroprotrophic thiab neurotrophic compound los ntawm inhibiting atp5a, tus tseem ceeb enzyme nyob rau hauv kev laus. Nws kuj tseem zoo li txhim kho kev tsim cov hlwb - derived neurotrophic factor (BDNF), uas pab neurons. Qhov cuam tshuam hauv tsiaj qauv: Tiv thaiv cov neurotoxicity hauv cov xovtooj ntawm tes. Txo cov qib amyloid - beta peptides thiab nce BDNF hauv cov hippocampus ntawm nas. Txhim kho cov nas. Tiv thaiv kev nco tsis nco qab hauv Alzheimer's - qauv mice. Qhia txog cov peev xwm rau lwm yam xwm txheej zoo li kev raug mob lub hlwb. |
Yuav ua li cas los tsim J 147 hmoov?
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Maj mam ntxiv trifluoroacetic anhydride herdride (0.33ml, 2.36g, 1.97mmide (0.33ml, 2.36mm) hauv dichhlorometomethane (5ml) ntawm 0℃thiab nyob rau hauv nitrogen tiv thaiv. Cov tshuaj tiv thaiv sib xyaw tau raug ntsia tsis tu ncua ntawm 0℃rau 1.5 teev. Tom qab cov tshuaj tiv thaiv tau ua tiav, cov sib xyaw kom muaj zog, thiab cov seem yog huv si los ntawm kem chromatography siv a (1:10) sib xyaw ua ke raws li cov khoom lag luamJ 147 hmoov(571 mg, tawm los 83%). |
Yuav ua li cas thiab qhov twg yuav J 147 hmoov?
Peb muaj 8 xyoo kev paub hauv kev muag cov tshuaj tshawb fawb txog kev cai lij choj thiab muaj lub koob npe zoo, ua rau peb tus khub uas ntseeg siab.
Peb paub tseeb tias qhov zoo ntawm peb cov khoom los ntawm kev sim ua haujlwm ywj pheej, thiab txhua tus neeg siv khoom yog peb VIP.
Xa koj qhov kev nug kom paub ntau ntxiv, Nyem Email:sales1@faithfulbio.comTam sim no.





Ntau hom kev xa khoom rau koj xaiv
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Tsheb Thauj Mus Los |
Shipping Txoj Kev |
Cargo Qhov hnyav |
Yam uas pab |
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3-7 hnub |
DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD, |
Haum rau hauv qab 50kg. |
Peb muaj cov chaw khaws khoom hauv Tebchaws Yelemees thiab California, Asmeskas, |
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7-15 hnub |
Los ntawm huab cua |
Haum rau ntau tshaj 50kg. |
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15-60 hnub |
Los ntawm hiav txwv |
Haum rau ntau tshaj 500kg. |
Cov FAQ
Q: Puas muaj kev phiv los ntawm J 147?
A: Lub siab bioavailability thiab ntshav - cov nyhuv rau nws cov kev cuam tshuam lub hlwb, tsis muaj ib qho tseem ceeb ntawm J147 tau tshaj tawm.
Q: Lub neej ntawm J 147 hmoov dab tsi?
A: (E / Z) - j147 ntsig txog cov tshuaj tiv thaiv kab mob
Ib nrab lub neej (t1/2) Ntawm (E / Z) {- J147 tau muab xam thaum 1.5 hrs hauv 1.5 teev hauv lub hlwb (PO) kev tswj hwm ntawm ib koob ntawm 20 mg / kg).
Q: J 147 nrhiav tau li cas?
A: J147 tau tsim kho xyoo 2011. J147 yog hloov kho version ntawm cov molecule (curcumin) pom nyob rau hauv curry Spice Turmeric.
Kev tsis lees paub: Cov lus ntawm lub vev xaib no yog siv rau kev tshawb fawb thiab kev kawm sib pauv. Thov ua tib zoo saib pom qhov tseeb ntawm lawv cov kev xav thiab cov ntsiab lus. Yog tias koj pom muaj kev ua txhaum. Thov hu rau tus thawj tswj hwm kom sai. Peb tsis yog lub luag haujlwm rau cov kev rau txim ntawm cov ntaub ntawv thiab cov kev pabcuam tau muab rau hauv lub vev xaib no.
Tsab ntawv: Cov khoom lag luam yog rau kev tshawb fawb tsuas yog siv thiab tsis yog rau kev kuaj mob, kev kho mob, tiv thaiv kab mob, thiab lwm yam.
Xa koj qhov kev nug kom paub meej ntxiv, nyem email:sales1@faithfulbio.comTam sim no.
Cim npe nrov: J 147 Hmoov CAS 1146963-51-0, Tuam Tshoj Tuam Tshoj, Cov Qauv, Kev Muag Khoom, Khoom Siv Dawb, Khoom Siv Raw, Ua Hauv Suav










