Oxcarbazepine hmoovyog prodrug. Nws yog ib qho qauv analogue ntawm 10- keto pawg ntawm carbamazepine, thiab feem ntau ntawm nws yog metabolized rau hauv active 10- hydroxy metabolites hauv vivo.
Oxcarbazepine hmoovyog ib qho 10- keto derivative ntawm carbamazepine, thiab nws cov txiaj ntsig zoo ib yam li lossis muaj zog me ntsis dua li ntawm carbamazepine. Carbamazepine thiab nws cov metabolites (hydroxyl derivatives) muaj cov tshuaj tiv thaiv kab mob thiab kev xaiv ntau yam inhibition ntawm cerebral cortex txav, uas tej zaum yuav yog vim thaiv qhov voltage-dependent sodium channel ntawm hlwb hlwb, yog li tiv thaiv kev sib kis ntawm focal paug. Tsis tas li ntawd, oxcarbazepine kuj ua rau cov poov tshuaj thiab calcium.
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| Cov duab tua tiag tiag ntawm Oxcarbazepine | Oxcarbazepine daim duab kos duab |
Khoom siv
1. Oxcarbazepine hmoovtuaj yeem thaiv qhov voltage-dependant sodium channels hauv hlwb hlwb,
2. Nws tuaj yeem ruaj khov ntawm cov paj hlwb overactive cell membrane,
3. Nws tuaj yeem inhibit qhov rov ua dua ntawm cov neurons,
4. Nws tuaj yeem txo qhov excitatory impulses kis los ntawm synapses.
Khoom Specification
Yam khoom | Specification | Cov txiaj ntsig |
Qhov tshwm sim | Ib tug dawb los yog yuav luag dawb, crystalline hmoov | Ua raws |
Kev txheeb xyuas | IR & UV & HPLC | Ua raws |
Solubility | Soluble hauv methanol thiab ethanol, insoluble hauv dej | Ua raws |
Melting point | 222 ~ 228 degree | 223 ~ 224 degree kub |
Poob rau ziab | Tsawg dua lossis sib npaug rau 0.3% | 0.21% |
Residue ntawm Ignition | Tsawg dua lossis sib npaug rau 0.2% | 0.09% |
txheeb ze yam khoom | Carbamazepine Tsawg dua lossis sib npaug rau 0.2% | 0.14% |
Tsis paub impurities Tsawg dua lossis sib npaug rau 0.5% | <0.5% | |
Tag nrho cov impurities Tsawg dua lossis sib npaug rau 1.0% | 0.54% | |
Assay | Ntau dua lossis sib npaug rau 99.0% | 99.56% |
Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:allen@faithfulbio.comTam sim no.
Koj tuaj yeem tiv tauj kuv ntawm WhatsApp:+86 13137770562





Muaj ntau txoj kev xa khoom rau koj xaiv
Tsheb thauj mus los | Shipping txoj kev | Cargo hnyav xav tau | Qhov zoo |
3-7 hnub | DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD, | Haum rau qis dua 50kg. | Peb muaj warehouses nyob rau hauv lub teb chaws Yelemees thiab California, lub teb chaws USA, |
7-15 hnub | Los ntawm Cua | Haum rau ntau tshaj 50kg. | |
15-60 hnub | Los ntawm Hiav Txwv | Haum rau ntau tshaj 500kg. |
Tsis lees paub: Cov ntawv luam tawm ntawm lub vev xaib no yog siv los txhawb kev sib pauv kev kawm thiab kev kawm, thiab tsis txhais hais tias lub vev xaib no pom zoo nrog nws cov kev xav lossis lees paub qhov tseeb ntawm nws cov ntsiab lus. Thov lim kom zoo. Yog tias koj ntseeg tias tsab xov xwm no ua txhaum, thov hu rau tus thawj tswj hwm. Peb tsis muaj lub luag haujlwm rau qhov tshwm sim ntawm kev siv cov ntaub ntawv thiab cov kev pabcuam hauv lub vev xaib no.
Nco tseg: Cov tshuaj no yuav tsum tau siv rau kev tshawb fawb nkaus xwb. Cov lus thov no tsis tau raug soj ntsuam los ntawm Food and Drug Administration. Thov nrog koj tus kws kho mob tham thiab kawm txog cov kev tshawb fawb muaj ua ntej siv lawv. Cov khoom no tsis yog tsim los kuaj xyuas, kho, kho lossis tiv thaiv kab mob.
Cim npe nrov: oxcarbazepine hmoov cas 28721-07-5, lwm tus neeg, manufacturers, hoobkas, lag luam wholesale, yuav, nqe, tej, ntshiab, tsim, kev muag khoom








