Khoom Piav Qhia

Carbetocin acetateyog cov khoom siv hluavtaws, tshwj xeeb ib txwm ua rau ntev-ua oxytocin analog, thiab muaj cov agonist muaj agonist ntawm Oxytocin receptor. Nws yog siv los tswj cov hemorrhates thiab los ntshav tom qab yug menyuam, tshwj xeeb yog tom qab Cesarean. Nws tau muaj kev ruaj khov ntau dua thiab ntev ntev ntawm kev ua piv rau oxytocin.
Carbetocin acetateyog kev txhim kho rau Oxytocin, uas tau txais kev hloov kho txheej txheem ntawm Oxytocin: (1) DEAMINATIONS, nrog rau pawg buloyl hloov ib CYS Oxytocin; (2) Disulfide Kev Ua Haujlwm: Txoj Haujlwm 4 ntawm cov pab pawg ByranicL ua qauv rau cov pab pawg thiaher rau ntawm lub sijhawm thib 6 ntawm Oxytocin Cys. (3) Hydroxyl Methylation ntawm Tyr. Cov kev hloov pauv saum toj saud tuaj yeem pab kom carbetocin acetate kom txo qis kev ua tsis raws cai ntawm cov enzymes thiab discfide sib txuas thiab txhim kho kev ruaj khov. Txawm hais tias muaj qhov sib txawv hauv lawv cov qauv molecular, lawv ib qho kev sib txawv rau cov khoom noj kom zoo nkauj hauv qhov myometrium yog tib yam. Vim kev hloov kho txheej txheem, qhov chaw ruaj khov ntawm carbetocin acetate yog muaj zog tshaj li Oxytocin.
Cov chaw kuaj mob thiab lub tsev muag tshuaj ntawm carbetocin acetate zoo ib yam li cov ntawm ib txwm ua oxytocin. Nws khi rau Oxytocin cov receptors hauv uterine du leeg, ua rau cov lus sib dhos ntawm lub tsev menyuam. Ntawm lub hauv paus ntawm thawj cov lus cog lus, nws nce ntau zaus thiab uterine nro. Hauv lub xeev tsis muaj cev xeeb tub, cov ntsiab lus ntawm Oxytocin cov receptors hauv lub tsev menyuam yog tsawg heev, nce thaum cev xeeb tub, thiab peaks thaum xa khoom. Yog li no, carbetocin acetate tsis muaj kev cuam tshuam rau lub tsev menyuam tsis muaj lub xeev xeeb tub, tab sis nws muaj cov lus cog lus rau lub tsev menyuam xeeb tub thiab lub tsev menyuam yog tom qab xa khoom.

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Coa
| lub ntsiab | Lub hom phiaj | Qho kawg |
| Kev piav txog | Dawb lossis yuav luag dawb hmoov | Ua raws |
| Hnyav Hlau | Tsawg dua los yog sib npaug rau 0.002% | Ua raws |
| Ywg dej | Tsawg dua los yog sib npaug ntawm 7.0% | 0.76% |
| Acetic acid cov ntsiab lus | Tsawg dua los yog sib npaug rau 12.0% | 6.20% |
| Kev coj dawb huv | Ntau dua los yog sib npaug rau 98.0% | 99.40% |
| Cov ntsiab lus ntawm Peptide | Ntau dua los yog sib npaug rau 80% | 92.10% |
| Ib Leeg Cav | Tsawg dua los yog sib npaug rau 1.0% | 0.12% |
| Tag | Ua raws li kev lag luam tshwj xeeb | |
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Quav: 1.2 ± 0.1 g / cm ³
Boint Taw tes: 1477.9 ± 650.0 Degree ntawm 760 MmHG
Molecular Cov Qauv: C45H69N11OOXS
Molecular hnyav: 988.161
Nyem Taw tes: 847.6 ± 34.3 Qib
Zoo heev Loj: 987.484802
PSA 387.81000
Logp -3.59
Carbetocin acetate ua dab tsi?
Carbetocin acetatePuas yog ib tus neeg sawv cev Oxytocin tau siv los tswj cov hemorrhates thiab los ntshav tom qab yug menyuam. Carbetocin yog yeeb tshuaj siv los tswj cov hemorrhage, los ntshav tom qab yug menyuam. Nws yog qhov analogue ntawm oxytocin, thiab nws cov kev txiav txim zoo ib yam li Oxytocin - nws ua rau lub koomhaum ntawm lub tsev menyuam.
Carbetocin puas tuaj yeem tiv thaiv tus tub ntxhais kawm ntawv hemorrhage?
Oxytocin ua haujlwm ntawm cov receptors ntawm cov leeg nqaij du thiab txhawb cov uterine sab saud los cog lus tsis tu ncua. Carbetocin yog ntev-ua hluavtaws oxytocin analogue thiab kuj ua haujlwm los ntawm kev txhawb nqa lub tsev menyuam. Muaj kev phiv zoo heev rau ob qho tshuaj, xws li xeev siab thiab ntuav.
Dab tsi yog qhov zoo ntawm carbetocin?
Carbetocin muaj cov txiaj ntsig dhau Oxytocin rau kev tiv thaiv ntawm tus menyuam kawm ntawv hemorrhatum. Piv nrog oxytocin, cua sov-ruaj khov carbetocin, tsis xav tau khaub thuas-saw thauj thiab cia.
Cov yam ntxwv tseem ceeb ntawm carbetocin acetate
Oxytocin receptor agonist: nws khi rau thiab ua kom ua kom oxytocin cov receptors, mimicking Oxytocin cov teebmeem.
Tom qab hemorrhage: nws yog siv los tiv thaiv thiab kho kom ntshav ntau dhau tom qab yug menyuam.
Ntev ntev ntawm kev nqis tes ua: carbetocin acetate muaj ib nrab ib nrab lub neej thiab muab cov nyhuv ntau dua li oxytocin.
Txhim kho cov khoom ruaj khov: nws ua rau muaj kev ruaj khov zoo nyob hauv vivo piv rau oxytocin.
Kev cuam tshuam ua piv txwv: nws tau pom tias tsim cov tshuaj tua kab-zoo li kev ua haujlwm ntawm kev ua haujlwm ntawm Oxytocin cov khoom siv hauv nruab nrab.
Xa koj qhov kev nug kom paub meej ntxiv, nyem email:sales4@faithfulbio.com

Vim li cas thiaj xaiv peb
Peb Lub Hoobkas


Lub thawv

Txoj kev xa khoom
|
Tsheb Thauj Mus Los |
Shipping Txoj Kev |
Cargo Qhov hnyav |
Yam uas pab |
|
3-7 hnub |
DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD, |
Haum rau hauv qab 50kg. |
Peb muaj cov chaw khaws khoom hauv Tebchaws Yelemees thiab California, Asmeskas, thiab cov neeg siv khoom hauv Tebchaws Europe thiab Asmeskas tuaj yeem txaus siab xa cov khoom ncaj qha los ntawm ob qhov chaw no. |
|
7-15 hnub |
Los ntawm huab cua |
Haum rau ntau tshaj 50kg. |
|
|
15-60 hnub |
Los ntawm hiav txwv |
Haum rau ntau tshaj 500kg. |
Xa koj qhov kev nug kom paub meej ntxiv, nyem email:sales4@faithfulbio.com
Cim npe nrov: carbetocin acetate CAS 37025-55-1, Tuam Tshoj, chaw tsim khoom, kev lag luam, khoom siv, khoom siv nyoos, ua nyob rau hauv Suav teb






