Levocetirizine dihydrochloride yog R-isomer ntawm Cetirizine dihydrochloride thiab ib tiam tshiab ntawm kev ua tau zoo heev uas tsis yog sedating antihistamines. Nws affinity rau H1 receptors yog ob zaug ntawm cetirizine hydrochloride, thiab cov koob tshuaj zoo yog ib nrab ntawm cetirizine hydrochloride. Cov txiaj ntsig kho mob tau pom tias nws muaj qhov zoo dua li loratadine, ebastine, Mizolastine, thiabFexofenadine. NtshiabLevocetirizine dihydrochloride USPyog ib tug dawb hygroscopic hmoov siv los kho raws caij nyoog allergic rhinitis, perennial allergic rhinitis, allergic conjunctivitis, chronic idiopathic urticaria, thiab lwm yam.
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Yam khoom |
SPECIFICATION |
TSEEM CEEB |
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CHARACTE RS
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Kev piav qhia |
DAWB RAU OB-WHITE POWDER |
OFF-WHTIE POWDER |
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SOUBILITY |
Dawb soluble nyob rau hauv dej, me ntsis soluble nyob rau hauv ISOpropanol thiab nyob rau hauv acetonitriLE |
CONFORM |
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IDENTIFICATION |
1) INFRARED ABSORPTION SPECTROPHOTOMETRY CORRESPONDS REFEREENCE Standard |
Kev sib haum xeeb |
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2) ULTRAVIOLE ABSORPTION SPECTROPHOTOMETRY CORRESIONS RAU COV Standard Standard |
Kev sib haum xeeb |
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3) Kev sim rau cov poov tshuaj yuav tsum yog qhov zoo |
C0NFORMS |
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Dej (KF) |
Tsawg dua los yog sib npaug rau 0.5% |
0.3% |
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HAIV NEEG |
Tsawg dua lossis sib npaug li 10PPM |
<10PPM |
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Cov khoom muaj feem xyuam (HPLC) |
Tus kheej impurity Tsawg dua lossis sib npaug rau 0.2% |
0.07% |
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Tag nrho impurity Tsawg dua lossis sib npaug rau 0.5% |
0.12% |
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RESIDUAL SOLVENTS (GC) |
CYCLOHEXANE Tsawg dua lossis sib npaug rau 1000PPM |
< LOQ(LOQ:50PPM) |
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ISOPROPANOL Tsawg dua lossis sib npaug rau 2000PPM |
178 ppm ua |
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ASSAY (HPLC) |
98.5%-101. |
100% |
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TEEB MEEM |
Ua raws li USP36 |
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Dab tsi yog qhov txawv ntawm cetirizine hydrochloride thiab Levocetirizine dihydrochloride?
Muaj qhov sib txawv ntawm cov qauv molecular thiab kev ua tau zoo ntawmLevocetirizine dihydrochloridethiab cetirizine hydrochloride.
1, Txawv molecular qauv:Cetirizine dihydrochloride yog ib daim ntawv racemic uas muaj ob sab laug-tes qauv thiab sab tes xis qauv; Cov khoom xyaw ntawm Levocetirizine dihydrochloride tsuas muaj cov qauv sab laug xwb. Cov txiaj ntsig tau pom tau tias cov qauv sab laug yog cov khoom muaj txiaj ntsig zoo ntawm cetirizine, nrog rau kev xaiv siab rau H1 receptors uas yog 30 npaug ntawm cetirizine. Nyob rau tib lub sijhawm, cov khoom no tsis muaj qhov tseem ceeb anticholinergic lossis los tiv thaiv serotonin, thiab nws cov nyhuv inhibitory hauv nruab nrab yog me me. Txawm li cas los xij, nws tuaj yeem cuam tshuam qhov sib txuam ntawm eosinophils. Tsim nyog siv cov khoom no yog txoj hauv kev kom tau txais txiaj ntsig zoo, xaiv, thiab kev sib tw peripheral H1 receptor antagonists.
2, Txawv pharmacological teebmeem:Raws li cov ntaub ntawv kev sim cuam tshuam, qhov kev sib khi muaj peev xwm ntawm levocetirizine hydrochloride rau tib neeg H1 histamine receptor yog 30 npaug ntawmCetirizine hydrochloride. Yog li ntawd, nyob rau tib koob tshuaj,Levocetirizine dihydrochloride USPmuaj cov nyhuv antihistamine muaj zog dua li Cetirizine dihydrochloride, thiab ua rau muaj kev phiv tshuaj txo qis. Tsis tas li ntawd, kev faib tawm thiab kev tswj hwm ntawm ob cov tshuaj no kuj txawv. Txawm li cas los xij, tsis hais txog qhov sib txawv ntawm lawv, nws yuav tsum sab laj nrog koj tus kws kho mob ua ntej thaum lub sijhawm tshawb fawb lossis kev siv theem.
Peb lub tuam txhab tuaj yeem muab Levocetirizine dihydrochloride, cetirizine hydrochloride, loratadine, ebastine, Mizolastine,Fexofenadinethiab lwm yam. ntawm tus nqi qis. Yog tias koj txaus siab, thov sau ntawv los ntawmemail:sales6@faithfulbio.com
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| 130018-87-0 Levocetirizine dihydrochloride | 83881-52-1 Cetirizine dihydrochloride | 90729-43-4 Ebastine | 83799-24-0 Fexofenadine |
Dab tsi yog qhov ua tau zoo thiab cov teebmeem ntawm levocetirizine hydrochloride ntsiav tshuaj?
Cov khoom tseem ceeb ntawm cov ntsiav tshuaj levocetirizine hydrochloride yog levocetirizine hydrochloride, uas yog siv los kho cov kab mob ua xua. Nws lub luag haujlwm tseem ceeb thiab cov teebmeem yog tiv thaiv kev ua xua, tiv thaiv khaus, tshem tawm urticaria, kho eczema, txhim kho mob hawb pob, thiab lwm yam. Nws raug nquahu kom siv cov tshuaj tshwj xeeb raws li kev qhia ntawm tus kws kho mob.
1. Antiallergy:Levocetirizine hydrochloride ntsiav tshuaj yog ib qho tshuaj tiv thaiv kab mob uas tuaj yeem cuam tshuam cov tshuaj histamine tso tawm, uas yog ib qho ntawm cov neeg kho mob tseem ceeb ua rau muaj kev tsis haum tshuaj.
2. Antipruritic:Los ntawm stabilizing mast cell membrane thiab txo qhov tso tawm ntawm nws sensitizing yam, lub hom phiaj ntawm relieving khaus yuav ua tau tiav.
3. Kho urticaria:Nws tuaj yeem txo cov tsos mob ntawm urticaria thiab tswj tus mob sai sai rau kev tawm tsam ntawm urticaria.
4. Kho eczema:xaiv antagonizing peripheral cov ntaub so ntswg H1 receptors, inhibiting mast cell degranulation, thiab tiv thaiv kev tso tawm ntawm inflammatory mediators muaj ib tug tej yam kev kho mob ntawm eczema.
5. Txhim kho mob hawb pob:Nws tuaj yeem cuam tshuam qhov kev tso tawm ntawm cov kab mob inflammatory mediators los ntawm mast hlwb, txo bronchial constriction thiab mucus secretion, yog li txhim kho txoj kev ua pa ntawm cov neeg mob hawb pob.
Tsis tas li ntawd, nws tuaj yeem txo cov tsos mob ntawm kev tsis haum rhinitis thiab allergic conjunctivitis. Thaum lub sij hawm siv cov ntshiab Levocetirizine dihydrochloride, nws yog ib qho tsim nyog yuav tsum tsis txhob tsav tsheb lub cev muaj zog lossis cov tshuab ua haujlwm kom tsis txhob muaj xwm txheej tshwm sim los ntawm kev tsis zoo xws li qaug zog. Cov tib neeg uas muaj keeb kwm ntawm daim siab ua haujlwm tsis zoo lossis tsis zoo yuav tsum siv ceev faj, thiab kev kho mob thiab kev txhawb nqa tau pom zoo tom qab noj ntau dhau. Tom qab noj cov tshuaj no, cov tshuaj tsis zoo xws li mob taub hau, tsaug zog, qhov ncauj qhuav, thiab qaug zog tuaj yeem tshwm sim. Yog tias cov tsos mob hnyav los yog tsis tu ncua, nws raug nquahu kom nrhiav kev kho mob sai.
Muaj ntau txoj kev xa khoom rau koj xaiv
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Tsheb thauj mus los |
Shipping txoj kev |
Cargo hnyav xav tau |
Qhov zoo |
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3-7 hnub |
DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD, |
Haum rau qis dua 50kg. |
Peb muaj warehouses nyob rau hauv lub teb chaws Yelemees thiab California, teb chaws USA, |
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7-15 hnub |
Los ntawm Cua |
Haum rau ntau tshaj 50kg. |
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15-60 hnub |
Los ntawm Hiav Txwv |
Haum rau ntau tshaj 500kg. |
Peb lub zog:
Peb lub tuam txhab tau dhau los ntawm FDA thiab ISO19001 kev tswj hwm qhov system ntawv pov thawj. Thiab peb muaj kev koom tes nrog kev cog lus nrog ntau lub chaw tsim khoom thiab chaw soj nstuam hauv Suav teb, Peb lub tuam txhab tuaj yeem muab Levocetirizine dihydrochloride, cetirizine hydrochloride, loratadine, ebastine, Mizolastine,Fexofenadinethiab lwm yam. ntawm tus nqi qis. Yog tias koj xav tau, thov sau ntawv
Peb tsis tsuas yog muaj qhov tshwj xeeb zoo hauv kev thauj mus los, tab sis kuj txhawb ntau txoj kev them nyiaj, txawm tias koj siv nyiaj US, euros, Australian las, lossis cov nyiaj hauv zos los ntawm Singapore, Malaysia, Thaib, thiab lwm yam. Peb kuj tuaj yeem txhawb cov txiaj ntsig hauv zos hauv cov cheeb tsam thiab cov tebchaws no. Tsis tas li ntawd, peb kuj txhawb nqa cov npav hauv txhab nyiaj (credit cards, thiab lwm yam) rau kev them nyiaj.
Tsis lees paub: Cov ntaub ntawv luam tawm ntawm lub vev xaib no los ntawm Is Taws Nem, tsis tau txhais hais tias lub vev xaib no pom zoo nrog nws cov kev xav lossis lees paub qhov tseeb ntawm cov ntsiab lus. Thov ua tib zoo saib kom paub qhov txawv. Tsis tas li ntawd, cov khoom muab los ntawm peb lub tuam txhab tsuas yog siv rau kev tshawb fawb tshawb fawb. Peb tsis muaj lub luag haujlwm rau qhov tshwm sim ntawm kev siv tsis raug.
Yog tias koj txaus siab rau peb cov khoom, lossis muaj cov lus qhia tseem ceeb ntawm peb cov khoom lossis tsis txaus siab rau cov khoom tau txais, thov hu rau peb los ntawmEmail :sales6@faithfulbio.com . Peb pab neeg tau cog lus los ua kom tiav kev txaus siab ntawm cov neeg siv khoom.
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