ATH-1017 CAS Nr .: 2093305-05-4

ATH-1017 CAS Nr .: 2093305-05-4

Khoom npe: ATH-1017
Lub ntsiab lus: Fosgonimeton; ATH-1017; Fosgonimeton (ATH-1017)
CAS Nr .: 2093305-05-4
EINECS NO.:/
Cov mis mos molecular: C27H45N4O8P
Purity & Qib: 99%; Qib tshuaj
Cim: Dawb hmoov
Cov qauv dawb: Muaj
Tshuag: Hauv Tshuag
Warehouse: USA/EU/AU Warehouse
MOQ & Pob: 1g; Pob raws li xav tau
Shipping: Kev nyab xeeb thiab xa khoom sai
Lub sij hawm xa tuaj: 7-15 hnub
Khw & Txee lub neej: Txias & qhuav qhov chaw; 24 hli
Xa kev nug
Hauj lwm lawm
 
 

Khoom piav qhia

Fosgonimeton

ATH-1017 CAS Nr .: 2093305-05-4yog ib tug zoo regulator (agonist) ntawm lub hepatocyte loj hlob yam (HGF)/c-Met receptor system. Nws tsis yog ib txwm peptide, tab sis me me molecule. HGF system plays lub luag haujlwm tseem ceeb hauv kev muaj sia nyob neuronal, synaptic plasticity, thiab kev kawm thiab kev nco.

Los ntawm kev ua kom cov kab ke no, Fosgonimeton aims los txhawb:

Neuroprotection: combating kev puas tsuaj los ntawm neurotoxicity, neuroinflammation, oxidative kev nyuaj siab, thiab excitotoxicity.

Neurotrophy: txhawb kev loj hlob ntawm neuronal, synapsis (tshiab synapse), thiab kev sib txuas neuronal.

Kev txhim kho kev txawj ntse: ua kom pom qhov cuam tshuam ntawm kev txhim kho kev txawj ntse hauv cov qauv ua ntej, tiv thaiv kev puas tsuaj los ntawm amyloid- (A) toxicity.

Txo Tau protein ntau hyperphosphorylation: lwm qhov tseem ceeb pathological ntawm Alzheimer tus kab mob.

Fosgonimeton peptide

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

COA

 

Cov khoom Specifications Cov txiaj ntsig
Qhov tshwm sim Dawb rau tawm -dawb hmoov Ua raws
Kev txheeb xyuas HNMR Conforms rau cov qauv Ua raws
LC-MS Conforms rau MW Ua raws
Poob rau ziab Tsawg dua lossis sib npaug li 1.0% 0.44%
Residue ntawm Ignition Tsawg dua los yog sib npaug li 0.5% 0.09%
Melting Point 174.0℃-181.0 degree 177.9℃-179.6 degree
Hnyav Hlau <10ppm <10ppm
Purity los ntawm HPLC Ntau dua lossis sib npaug li 99.0% 99.71%
Xaus Ua raws li kev lag luam specification

 

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MF of ATH-1017

Cov mis mos molecular: C27H45N4O8P
Molecular Luj: 584.64
Cia tej yam kev mob: -20 degree

 

R&D xwm txheej ntawm ATH-1017 CAS 2093305-05-4

 

ATH-1017 CAS 2093305-05-4 yog tam sim no nyob rau hauv kev sim tshuaj

Alzheimer's disease (AD): Ntau qhov kev sim tshuaj tau ua, suav nrog LIFT-AD (Phase II/III) thiab ACT-AD (Phase II pov thawj- ntawm- tswvyim) kev sim. Txawm li cas los xij, cov txiaj ntsig tsis ntev los no tau pom tias cov khoom lag luam ua tsis tau raws li qhov tseem ceeb lossis cov ntsiab lus tseem ceeb thib ob ntawm LIFT-AD mus sib hais. Yog li ntawd, txoj kev loj hlob rau qhov qhia txog tus kab mob Alzheimer's tau raug tso tseg.

Parkinson's disease dementia thiab Lewy lub cev dementia: Cov txiaj ntsig ntawm Phase II SHAPE sim qhia "txhawb" cov cim qhia, txhawb lub peev xwm kho lub luag haujlwm ntawm kev tswj hwm zoo ntawm HGF system hauv cov kab mob no, tab sis txoj kev loj hlob ntawm qhov taw qhia tam sim no kuj pom tias raug ncua.

Cov ntsiab lus

Fosgonimeton yog ib qho khoom lag luam me me uas muaj lub hom phiaj los daws cov kab mob nyuaj ntawm ntau yam kab mob neurodegenerative los ntawm kev tsom mus rau HGF/c-Met neurotrophic system. Txawm hais tias muaj kev txhawb nqa cov ntaub ntawv preclinical, cov ntsiab lus tseem ceeb ntawm kev ua tau zoo tsis tau ua tiav nyob rau hauv qhov tseem ceeb lig - kev sim tshuaj rau Alzheimer's kab mob thiab Lewy lub cev dementia. Tam sim no, nws txoj kev kho mob rau cov kev qhia no tau raug ncua.

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

ATH-1017 CAS 2093305-05-4

vim li cas xaiv peb

 
Peb ua raws li lub hauv paus ntsiab lus ntawm "cov neeg siv khoom ua ntej, kev ua siab ncaj ua ntej", thiab ib txwm muab cov neeg siv khoom nrog cov khoom zoo thiab muaj txiaj ntsig zoo thiab siab - cov kev pabcuam zoo. Xaiv kev ntseeg. Xaiv lub neej noj qab nyob zoo!
 
Nrog rau peb cov kev siv zog tas mus li thiab kev pabcuam zoo, peb cia siab tias yuav tsim kom muaj kev koom tes ntev - thiab kev loj hlob zoo nrog cov neeg siv khoom thiab muab sijhawm rau peb. Peb ntseeg tias peb yuav ua rau koj txaus siab rau thawj -chav kawm zoo, nyab xeeb thiab xa khoom sai thiab txaus siab tom qab- kev muag khoom.

 

Peb lub Hoobkas

 

ATH-1017 CAS 2093305-05-4

ATH-1017 CAS 2093305-05-4

 

Pob

 

ATH-1017 CAS 2093305-05-4

 

Shipping Txoj Kev

 

Tsheb thauj mus los

Shipping txoj kev

Cargo hnyav xav tau

Qhov zoo

3-7 hnub

DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD,
UPS, USPS, FedEx, TNT, EMS

Haum rau qis dua 50kg.
International qhov rooj rau qhov rooj nthuav qhia

Peb muaj warehouses nyob rau hauv lub teb chaws Yelemees thiab California, teb chaws USA, thiab cov neeg muas zaub nyob rau hauv cov teb chaws Europe thiab America muaj peev xwm txaus siab rau xa cov khoom ncaj qha los ntawm ob qhov chaw.

7-15 hnub

Los ntawm Cua

Haum rau ntau tshaj 50kg.
ceev thiab pheej yig dua rau kev txiav txim loj

15-60 hnub

Los ntawm Hiav Txwv

Haum rau ntau tshaj 500kg.
Kev xa khoom pheej yig tshaj plaws

 

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

 

FAQ

 

 

01. Dab tsi yog ATH-1017 CAS 2093305-05-4? Puas yog peptide?

Fosgonimeton (ATH-1017) yog ib qho me me molecule prodrug uas tau hloov pauv sai hauv vivo rau hauv cov metabolite fosgo-AM (ATH-1001). Nws tsis yog ib qho khoom peptide nyob rau hauv kev xav ib txwm.

02. Lub tshuab ua haujlwm ntawm ATH-1017 CAS 2093305-05-4 yog dab tsi?

Nws cov txheej txheem tseem ceeb ntawm kev ua haujlwm yog qhov kev hloov pauv ntawm cov kab mob hepatocyte loj hlob (HGF)/c-Met signaling system. Txoj kev taw qhia no tuaj yeem cuam tshuam rau cov kab mob neurodegenerative. Los ntawm kev txhim kho cov kab ke no, Fosgonimeton lub hom phiaj los muab kev tiv thaiv neuroprotection, txhawb kev noj qab haus huv neuronal thiab kev ciaj sia, tiv thaiv synaptic networks, thiab muaj kev cuam tshuam los tiv thaiv -, yog li muaj peev xwm ua rau qeeb ntawm cov kab mob neurodegenerative thiab txhim kho kev txawj ntse. Hauv cov qauv ua ntej, nws tau pom tias muaj kev tawm tsam amyloid - (A ) toxicity, txo tau protein ntau hyperphosphorylation, thiab txhim kho kev txawj ntse.

03. Kev nyab xeeb npaum li cas ATH-1017 CAS 2093305-05-4?

Hauv kev sim tshuaj,ATH-1017 CAS Nr .: 2093305-05-4feem ntau pom zoo rau kev zam thiab kev nyab xeeb.
 
Tsis lees paub: Tag nrho cov khoom lag luam (tsis yog- cov khoom raug cai) cov duab raug coj los ua zoo, tab sis vim yog lub zog ntawm lub teeb (lub sijhawm sib txawv, lub teeb tom qab sib txawv), cov txheej txheem tua, cov khoom siv sib txawv thiab lwm yam, tej zaum yuav muaj qee qhov sib txawv ntawm daim duab thiab cov xim tiag tiag, cov xim ntawm cov khoom, thov coj cov nyhuv tiag tiag, xim txawv ntawm cov khoom tsis yog qhov teeb meem zoo.
 
Nco tseg: Nco ntsoov sab laj nrog tus kws kho mob uas tsim nyog ua ntej noj cov tshuaj tshiab. Cov khoom no tsis yog tsim los kuaj xyuas, kho, kho lossis tiv thaiv txhua yam kab mob.Thaum lub sijhawm yuav khoom, tus neeg yuav khoom thoob ntiaj teb pom zoo xav tias muaj kev pheej hmoo ntawm txhua yam khoom tuaj txog. Peb tsis tuaj yeem hloov cov khoom ploj lossis raug kaw. Ua ntej xa cov khoom, koj yuav tsum paub meej tias koj pom zoo rau cov nqe lus no.Qhov no tsuas yog kev pom zoo koob tshuaj raws li peb tus kheej kev paub thiab cov ntaub ntawv pov thawj. Peb pom zoo kom koj ua koj tus kheej kev tshawb fawb ua ntej siv cov khoom no.
 
Nqe lus:Cov khoom no tsuas yog siv rau kev tshawb fawb tshawb fawb, thiab qhov tshwm sim ntawm lwm yam kev siv tsis muaj lub luag haujlwm.

 

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