Formoterol Fumarate Dihydrate API CAS 183814-30-4

Formoterol Fumarate Dihydrate API CAS 183814-30-4

Khoom npe: Formoterol fumarate dihydrate API
CAS Nr .: 183814-30-4
Cov mis mos molecular: C23H28N2O8
EINECS.NO:/
Lub ntsiab lus: Formoterol fumarate dihydrate; Unii-W34shf8J2k; Formoterol fumarate dihydrate, 98.5%; Formoterol Fumarate (100 mg); forMaMide fuMarate dihydrate
Test Method: HPLC/UV
MOQ & Pob: 10g, 100g, 1kg thiab lwm yam Sub- pob
Daim ntawv pov thawj: FDA, ISO, COA, HPLC, MSDS, TDS thiab lwm yam
Lub Sijhawm Lead: 1-3 hnub
Shipping: DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD, UPS, USPS, FedEx, EMS, Los ntawm Cua, Los ntawm hiav txwv thiab lwm yam
Khw & Txee lub neej; Txias & qhuav qhov chaw; 36 lub hlis
Lwm yam: Muaj warehouses nyob rau hauv lub tebchaws United States, Australia thiab lub teb chaws Yelemees.
Xa kev nug
Hauj lwm lawm

Formoterol fumarate dihydrate yog dab tsi?

Formoterol hemifumarate hydrate tsis yog tsuas yog xaiv, ntev - ua 2-adrenergic receptor agonist, tab sis kuj yog ntev - ua bronchodilator siv hauv kev tshawb fawb txog kev mob hawb pob thiab mob ntsws ntsws ntev. Nws relaxes cov nqaij ntshiv nyob ib ncig ntawm cov pa, tso cai rau cov pa ib ntsuj av tau rov qhib dua. Nws qhov tseem ceeb tshaj plaws yog nws "dual effect": qhov pib sai thiab siv tau ntev.Formoterol fumarate dihydrate APItseem tuaj yeem ua rau mitochondrial biogeneration tom qab mob hlwb thiab txhawb kev paub txog kev rov qab los.

Yog li ntawd, nws tuaj yeem siv rau kev kho mob niaj hnub thiab, raws li kws kho mob cov lus qhia, rau kev tiv thaiv kev tawm dag zog -ua rau mob plab.

tiv tauj peb ntawm Email :sales6@faithfulbio.com

 

Yuav ua li cas yog lub mechanism ntawm kev txiav txim ntawm Formoterol fumarate dihydrate?

Formoterol fumarate dihydrate feem ntau ua raws li cov receptors tshwj xeeb ntawm cov leeg hauv cov hlab ntsha, pib ua cov txheej txheem sib kis hauv lub cev. Thaum cov khoom khi khi rau cov receptor, nws yuav txhawb kev hloov pauv ntawm cov khoom muaj feem xyuam hauv lub cev, qhib cov tshuaj nquag, maj mam txo cov calcium ion cov ntsiab lus hauv cov hlab ntsws, tso cai rau cov leeg mob ntsws kom maj mam so, qhib txoj hlab pa, thiab yooj yim alleviating ua pa nyuaj.
Cov khoom siv raw no muaj zog lipid solubility thiab tuaj yeem ua raws thiab nyob twj ywm rau hauv cov pa cell membrane kom qeeb tso tawm. Nws tuaj yeem siv tau sai sai li ntawm ob peb feeb tom qab nqus tau thiab tuaj yeem muab cov nyhuv ruaj khov ntev txog li kaum ob teev tom qab siv ib zaug. Nws yuav siv sij hawm rau hauv tus account ob qho tib si ceev thiab qeeb cuam tshuam.
Nyob rau hauv cov lus pom zoo, nws tsuas yog tsom mus rau dilate thiab tshem tawm txoj hlab pa, tsis zoo li yuav ua rau lub cev tsis muaj zog, thiab cov nyhuv ntawm cov tshuaj kuj tseem tuaj yeem tswj xyuas kom ntev ntev ntawm kev siv. Tsis tas li ntawd, nws tuaj yeem tswj hwm ntau txoj hauv kev physiological hauv lub cev, pab ua kom cov cell metabolism hauv ib txwm muaj, thiab txo qis kev tso tawm cov tshuaj inflammatory hauv lub cev. Nws tsis tsuas yog tshem tawm txoj kev ua pa xwb tab sis kuj muaj ntau yam haujlwm xws li soothing thiab tswj, thiab kho cov kab mob ua pa.
Zuag qhia tag nrho, nws tso siab rau lub hom phiaj meej, ntev - ua raws li kev txhawb nqa - tso tawm cov yam ntxwv, cov yam ntxwv me me thiab tsis kam rau siab, nrog rau ntau yam cuam tshuam xws li pab tiv thaiv - mob thiab kho, tsim kom muaj kev ua pa zoo thiab ruaj khov ua rau cov kab mob ua pa.

The mechanism of action of Formoterol fumarate dihydrate

 

Vim li cas Formoterol fumarate dihydrate ua haujlwm nrawm thiab kav ntev?

Superiority of Formoterol Fumarate Dihydrate

Formoterol fumarate (100 mg) ua tiav ob qho tib si pib sai thiab ntev - kev ua haujlwm ntev heev vim nws cov qauv molecular ntaus ib qho kev sib npaug zoo ntawm hydrophilicity thiab lipophilicity. Nws qhov pib sai yog vim nws qhov zoo tshaj hydrophilicity; tsis zoo li cov khoom lipophilic uas yuav tsum tau ua ntej diffuse tom qab rau hauv daim nyias nyias,Formoterol fumarate dihydrate APIdiffuses sai sai ncaj qha los ntawm aqueous theem ntawm cov pa tom qab nqus tau pa, khi rau lub orthotropic binding qhov chaw ntawm 2 receptors nyob rau hauv lub cell membrane nto, yog li tsis txhob ncua sij hawm pib. Nws lub sijhawm ntev ntawm kev ua haujlwm yog vim nws qhov zoo lipophilicity: nws cov molecules tuaj yeem nyob ib ntus nyob rau hauv cov lipid txheej ntawm cov hlab ntsha hauv cov hlab ntsha, tsim cov chaw cia, thiab tom qab ntawd maj mam tso tawm kom tsis tu ncua ua rau lub hom phiaj ntawm qhov chaw; Ntxiv mus, nws qeeb dissociation tom qab khi rau lub receptor tso cai rau lub sij hawm ntev ntawm kev txiav txim nrog txhua qhov khi. Qhov sib npaug ntawm qhov sib npaug ntawm hydrophilicity thiab lipophilicity ua rau formoterol fumarate dihydrate nkaus xwb - ua, ntev - kav ntev 2 agonist tam sim no muaj uas sib txuas qhov pib sai thiab ruaj khov - tso tawm cov khoom ntawm cov tshuaj thaum muaj xwm ceev.

 

MF ntawm Formoterol fumarate dihydrate

Molecular hnyav 460.48
Melting point 116-120 degree
Solubility DMSO: soluble, 20 mg/mL
Flash point 318.6 degree
MF Of Formoterol Fumarate Dihydrate

 

Specification

Yam khoom Specification Kev tshwm sim
Qhov tshwm sim Dawb rau tawm -dawb Ua raws
Dej (KF) 4.0~5.0% 4.20%
Sulphate tshauv Tsawg dua lossis sib npaug li 0.1% 0.04%
Cov hlau hnyav Tsawg dua lossis sib npaug li 20ppm Ua raws
Assay Ntau dua lossis sib npaug li 98.5% 99.40%
Xaus Ua raws li kev lag luam specification

 

Muaj ntau txoj kev xa khoom rau koj xaiv

Tsheb thauj mus los

Shipping txoj kev

Cargo hnyav xav tau

Qhov zoo

3-7 hnub

DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD,
UPS, USPS, FedEx, TNT, EMS

Haum rau qis dua 50kg.
International qhov rooj rau qhov rooj nthuav qhia

Peb muaj warehouses nyob rau hauv lub teb chaws Yelemees thiab California, teb chaws USA,
thiab cov neeg siv khoom hauv Tebchaws Europe thiab Asmeskas tuaj yeem
txaus siab xa khoom ncaj qha los ntawm ob qhov chaw no.

7-15 hnub

Los ntawm Cua

Haum rau ntau tshaj 50kg.
ceev thiab pheej yig dua rau kev txiav txim loj

15-60 hnub

Los ntawm Hiav Txwv

Haum rau ntau tshaj 500kg.
Kev xa khoom pheej yig tshaj plaws

 

Peb lub zog:

Peb lub tuam txhab tau dhau los ntawm FDA thiab ISO19001 kev tswj hwm qhov system ntawv pov thawj. Thiab peb muaj kev koom tes nrog kev cog lus nrog ntau lub Hoobkas thiab chaw kuaj hauv Suav teb, Peb lub tuam txhab tuaj yeem muabFormoterol fumarate dihydrate APIthiab lwm yam ntawm tus nqi zoo dua. Yog tias koj txaus siab, thov sau ib tsab ntawv.
Peb tsis tsuas yog muaj qhov tshwj xeeb zoo hauv kev thauj mus los, tab sis kuj txhawb ntau txoj kev them nyiaj, txawm tias koj siv nyiaj US, euros, Australian las, lossis cov nyiaj hauv zos los ntawm Singapore, Malaysia, Thaib, thiab lwm yam. Peb kuj tuaj yeem txhawb cov txiaj ntsig hauv zos hauv cov cheeb tsam thiab cov tebchaws no. Tsis tas li ntawd, peb kuj txhawb nqa cov npav hauv txhab nyiaj (credit cards, thiab lwm yam) rau kev them nyiaj.

 

FAQ:

Q1: Dab tsi yog qhov zoo ntawm Formoterol fumarate dihydrate's "dual-effect" ua ke?
Nws qhov tshwj xeeb tshaj plaws yog nws "dual-kev sib xyaw ua ke": nws siv tau sai heev, ua haujlwm tsis pub dhau 1-3 feeb ntawm kev nqus pa, thaum tseem muab cov teebmeem ntev, nrog rau ib daim ntawv thov ntev txog 12 teev.
Q2: Formoterol fumarate dihydrate puas tuaj yeem siv ib leeg rau ntev - kho mob hawb pob?
Cov neeg mob hawb pob yuav tsum tsis txhob siv Formoterol Fumarate (100 mg) ib leeg, vim nws tuaj yeem ua rau lawv cov mob hnyav zuj zus tuaj thiab muaj kev pheej hmoo siab heev. Cov neeg mob COPD tuaj yeem siv nws ib leeg rau kev saib xyuas thiab kev tswj hwm raws li kev qhia ntawm tus kws kho mob.
Q3: Dab tsi yog qee qhov kev phiv tshwm sim uas yuav tshwm sim tom qab siv Formoterol fumarate dihydrate?

Tej yam tshwm sim tsis zoo rauFormoterol fumarate dihydrate APIsuav nrog qhov ncauj qhuav, palpitations, tshee (tshwj xeeb tshaj yog nyob rau hauv tes), thiab mob taub hau. Cov tshuaj tiv thaiv no muaj feem xyuam rau 2 receptor agonism thiab feem ntau yog tshaj tawm thaum ntxov. Cov neeg mob feem ntau tuaj yeem zam tau lawv lub sijhawm, tab sis yog tias mob hnyav heev, yuav tsum tau nrhiav kev kho mob tam sim ntawd.

 

Tsis lees paub: Cov ntaub ntawv luam tawm ntawm lub vev xaib no los ntawm Is Taws Nem, tsis tau txhais hais tias lub vev xaib no pom zoo nrog nws cov kev xav lossis lees paub qhov tseeb ntawm cov ntsiab lus. Thov ua tib zoo saib kom paub qhov txawv. Tsis tas li ntawd, cov khoom muab los ntawm peb lub tuam txhab tsuas yog siv rau kev tshawb fawb tshawb fawb. Peb tsis muaj lub luag haujlwm rau qhov tshwm sim ntawm kev siv tsis raug.

Yog tias koj txaus siab rau peb cov khoom, lossis muaj cov lus qhia tseem ceeb ntawm peb cov khoom lossis tsis txaus siab rau cov khoom tau txais, thov hu rau peb los ntawmEmail :sales6@faithfulbio.com . Peb pab neeg tau cog lus los ua kom tiav kev txaus siab ntawm cov neeg siv khoom.

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