Khoom piav qhia

Rov qab transcriptase inhibitors
Nevirapineyog thawj zaug pom zoo tsis-nucleoside thim rov qab transcriptase inhibitor, ua raws li delavirdine. Nevirapine yog siv ua ke nrog lwm cov tshuaj tiv thaiv kab mob rau kev kho HⅣ-1 kab mob. Cov tshuaj no ib leeg yuav sai sai tsim cov kab mob resistant tib yam. Yog li ntawd, nevirapine yuav tsum ib txwm siv ua ke nrog tsawg kawg ob lwm yam tshuaj tiv thaiv kab mob.
Action mechanism
Nevirapinekhi ncaj qha rau qhov rov qab transcriptase ntawm HIV-1 thiab thaiv cov haujlwm ntawm RNA-dependent thiab DNA-dependent DNA polymerase los ntawm kev rhuav tshem cov catalytic site ntawm cov enzyme.
Kev ua si lom neeg
Nevirapine (NSC 641530) yog non-nucleoside reverse transcriptase inhibitor (NNRTI) rau kev kho mob HIV-1 kab mob thiab AIDS.
Cov cuab yeej tshuaj
Crystallization los ntawm pyridine - dej, melting point 247-249 degree . npo 2.8. Lipophilic; Distribution coefficient 83. Hanish degree hauv dej: txog 0.1mg/ml(Ph neutral); Soluble ntawm Ph <3.
siv
Nevirapine yog ib qho kev thim rov qab transcriptase inhibitor antiviral siv hauv kev kho mob AIDS.

Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com
COA
| Cov khoom kuaj | Specifications | Cov txiaj ntsig | |
| Cov cim | Kev piav qhia | Dawb mus rau dawb, tsis muaj ntxhiab mus ze li odorless, crystalline hmoov. | Tawm-dawb, tsw ntxhiab, crystalline hmoov |
| Solubility | Me ntsis soluble, xyaum insoluble hauv dej. | Ua raws | |
| Kev txheeb xyuas | A: Lub sijhawm khaws cia ntawm lub ncov loj hauv chromatogram ntawm Assay kev npaj sib raug rau qhov hauv chromatogram ntawm Kev Npaj Txuj Ci, raws li tau txais hauv Assay. | Ua raws | |
| B: Infrared absorption spectrophotometry: sib raug rau tus qauv siv. | Ua raws | ||
| Dej | Tsawg dua lossis sib npaug rau 0.2% | <0.1% | |
| Residue ntawm ignition | Tsawg dua lossis sib npaug rau 0.1% | <0.1% | |
| Cov hlau hnyav | Tsawg dua lossis sib npaug rau 0.001% | <0.001% | |
| Yam khoom (HPLC) | lmpurity A Tsawg dua lossis sib npaug rau 0.2% | N.D | |
| lmpurity B Tsawg dua lossis sib npaug rau 0.2% | <> | ||
| lmpurity C Tsawg dua lossis sib npaug rau 0.2% | <> | ||
| Lwm tus neeg uas tsis tau teev meej impurity Tsawg dua lossis sib npaug rau 0.1% | 0.07% | ||
| Tag nrho impurities Tsawg dua lossis sib npaug rau 0.6% | 0.07% | ||
| Kev ntsuam xyuas (HPLC) | 98. | 99.72% | |
| Residual solvents (GC) | Ethanol Tsawg dua lossis sib npaug li 3000ppm | N.D | |
| Xaus | Ua raws li kev lag luam specification | ||
Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com
Dab tsi yog qhov txawv ntawm nevirapine thiab efavirenz?
Nevirapine metabolism yog rhiab heev rau induction ntawm hepatic enzymes tshaj li ntawm Efavirenz; Yog li ntawd, Efavirenz-raws li kev tswj hwm tau tawm tswv yim los ua thawj kab kev kho mob hauv cov neeg mob HIV-TB.
Nevirapine controversy yog dab tsi?
Kev siv nevirapine los tiv thaiv kev sib kis ntawm niam mus rau tus menyuam tau muaj teeb meem. Kev thov ntawm cov tshuaj toxicity siab tsis tau lees paub hauv kev sim tshuaj lossis kev pabcuam dav dav ntawm kev siv cov txheej txheem.
Yam tshuaj twg yog nevirapine?
Nevirapine yog nyob rau hauv ib chav kawm ntawm cov tshuaj hu ua non-nucleoside reverse transcriptase inhibitors (NNRTIs). Nws ua haujlwm los ntawm kev txo qis tus kabmob HIV hauv cov ntshav.
Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com

vim li cas xaiv peb
Peb lub Hoobkas


Pob

Shipping Txoj Kev
|
Tsheb thauj mus los |
Shipping txoj kev |
Cargo hnyav xav tau |
Qhov zoo |
|
3-7 hnub |
DHL, Lub teb chaws Yelemees DHL, Lub teb chaws Yelemees DPD, |
Haum rau qis dua 50kg. |
Peb muaj warehouses nyob rau hauv lub teb chaws Yelemees thiab California, teb chaws USA, thiab cov neeg muas zaub nyob rau hauv cov teb chaws Europe thiab America yuav txaus siab rau xa cov khoom ncaj qha los ntawm ob qhov chaw. |
|
7-15 hnub |
Los ntawm Cua |
Haum rau ntau tshaj 50kg. |
|
|
15-60 hnub |
Los ntawm Hiav Txwv |
Haum rau ntau tshaj 500kg. |
Xa koj Cov Lus Nug kom paub meej ntxiv, Nyem email:sales4@faithfulbio.com
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